Adenylate cyclase agonist properties of CGP-12177A in brown fat: evidence for atypical beta-adrenergic receptors (Q68292807)

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23 September 2019

title

Adenylate cyclase agonist properties of CGP-12177A in brown fat: evidence for atypical beta-adrenergic receptors (English)

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23 September 2019

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ChEBI release 2020-05-28

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https://api.crossref.org/works/10.1152/AJPENDO.1991.260.2.E226

25 October 2022

author name string

P. J. Scarpace

1

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25 October 2022

M. Matheny

2

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language of work or name

English

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publication date

1 February 1991

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full work available at URL

23 September 2019

https://www.physiology.org/doi/pdf/10.1152/ajpendo.1991.260.2.E226

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American Journal of Physiology

25 October 2022

published in

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23 September 2019

volume

260

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23 September 2019

issue

2 Pt 1

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23 September 2019

page(s)

E226-31

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The brown adipocyte beta-adrenoceptor

23 September 2019

cites work

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A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

25 October 2022

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

25 October 2022

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25 October 2022

Molecular Pharmacology

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DE LEAN A., A.

1982

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Molecular characterization of the human beta 3-adrenergic receptor

25 October 2022

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(+/-)[125Iodo] cyanopindolol, a new ligand for beta-adrenoceptors: identification and quantitation of subclasses of beta-adrenoceptors in guinea pig.

25 October 2022

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Molecular Pharmacology

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ENJALBERT A., M.

1978

1 reference

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Brown adipose tissue metabolism and thermogenesis

25 October 2022

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25 October 2022

Molecular Pharmacology

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KENT R. S.

1980

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Direct assessment of beta-adrenergic receptors in intact rat adipocytes by binding of [3H]CGP 12177. Evidence for agonist high-affinity binding complex and for beta 1 and beta 2 receptor subtypes

25 October 2022

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The beta-adrenergic radioligand [3H]CGP-12177, generally classified as an antagonist, is a thermogenic agonist in brown adipose tissue

25 October 2022

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Comparison of the pharmacological profiles of adrenergic drugs (including BRL-agonists) at [3H]prazosin and [3H]CGP-12177 binding sites in brown adipose tissue

25 October 2022

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https://api.crossref.org/works/10.1152/AJPENDO.1991.260.2.E226

Age-associated decrease of adenylate cyclase activity in rat myocardium

25 October 2022

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Beta-adrenergic agonist-mediated desensitization in senescent rats

25 October 2022

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Molecular mechanisms of receptor desensitization using the beta-adrenergic receptor-coupled adenylate cyclase system as a model

25 October 2022

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https://api.crossref.org/works/10.1152/AJPENDO.1991.260.2.E226

25 October 2022

Identifiers

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23 September 2019

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