Modelling study of protein kinase inhibitors: binding mode of staurosporine and origin of the selectivity of CGP 52411 (Q71491544)

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19 October 2019

title

Modelling study of protein kinase inhibitors: binding mode of staurosporine and origin of the selectivity of CGP 52411 (English)

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19 October 2019

author name string

P Furet

1

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19 October 2019

G Caravatti

2

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19 October 2019

N Lydon

3

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19 October 2019

J P Priestle

4

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19 October 2019

J M Sowadski

5

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19 October 2019

U Trinks

6

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19 October 2019

P Traxler

7

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19 October 2019

publication date

1 December 1995

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Journal of Computer - Aided Molecular Design

19 October 2019

published in

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19 October 2019

volume

9

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19 October 2019

issue

6

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19 October 2019

page(s)

465-472

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Dianilinophthalimides: potent and selective, ATP-competitive inhibitors of the EGF-receptor protein tyrosine kinase

19 October 2019

cites work

1 reference

12 December 2020

Crystal structure of the catalytic subunit of cAMP-dependent protein kinase complexed with MgATP and peptide inhibitor

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12 December 2020

Inhibitors of protein kinase C. 3. Potent and highly selective bisindolylmaleimides by conformational restriction

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Crystal structure of the tyrosine kinase domain of the human insulin receptor

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12 December 2020

A new alkaloid AM-2282 OF Streptomyces origin. Taxonomy, fermentation, isolation and preliminary characterization

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RETRACTED: 4,5-Dianilinophthalimide: a protein-tyrosine kinase inhibitor with selectivity for the epidermal growth factor receptor signal transduction pathway and potent in vivo antitumor activity

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12 December 2020

Predictor for sulfur-aromatic interactions in globular proteins

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12 December 2020

Signal-transduction therapy. A novel approach to disease management

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12 December 2020

Assignment of conserved amino acid residues to the ATP site in the protein kinase domain of the receptor for epidermal growth factor

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12 December 2020

Characterization of receptor tyrosine-specific protein kinases by the use of inhibitors. Staurosporine is a 100-times more potent inhibitor of insulin receptor than IGF-I receptor.

1 reference

12 December 2020

Structural features that specify tyrosine kinase activity deduced from homology modeling of the epidermal growth factor receptor

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12 December 2020

Structure of a peptide inhibitor bound to the catalytic subunit of cyclic adenosine monophosphate-dependent protein kinase

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12 December 2020

A new inhibitor of protein kinase C, RK-286C (4'-demethylamino-4'-hydroxystaurosporine). I. Screening, taxonomy, fermentation and biological activity.

1 reference

12 December 2020

The protein kinase family: conserved features and deduced phylogeny of the catalytic domains

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12 December 2020

Crystal structure of casein kinase-1, a phosphate-directed protein kinase

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12 December 2020

Atomic structure of the MAP kinase ERK2 at 2.3 A resolution

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12 December 2020

Characterization of specific binding sites for [3H]-staurosporine on various protein kinases

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12 December 2020

Crystal Structure of the Catalytic Subunit of Cyclic Adenosine Monophosphate-Dependent Protein Kinase

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12 December 2020

Phosphotransferase and substrate binding mechanism of the cAMP-dependent protein kinase catalytic subunit from porcine heart as deduced from the 2.0 A structure of the complex with Mn2+ adenylyl imidodiphosphate and inhibitor peptide PKI(5-24)

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12 December 2020

Two structures of the catalytic domain of phosphorylase kinase: an active protein kinase complexed with substrate analogue and product

1 reference

12 December 2020

Crystal structure of cyclin-dependent kinase 2

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12 December 2020

Inhibitors of protein kinase C. 2. Substituted bisindolylmaleimides with improved potency and selectivity

1 reference

12 December 2020

Staurosporine, a potent inhibitor of phospholipid/Ca++dependent protein kinase

1 reference

12 December 2020

Identifiers

DOI

10.1007/BF00124317

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8789188%20AND%20SRC:MED&resulttype=core&format=json

journals/jcamd/FuretCLPSTT95

19 October 2019

DBLP publication ID

1 reference

DBLP Dataset 2021-01-02

28 January 2021

1 reference