Probing the V1a vasopressin receptor binding site with pyroglutamate-substituted linear antagonists (Q71678974)

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20 October 2019

title

Probing the V1a vasopressin receptor binding site with pyroglutamate-substituted linear antagonists (English)

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20 October 2019

4

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20 October 2019

author name string

J Howl

series ordinal

1

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20 October 2019

N J Yarwood

series ordinal

2

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20 October 2019

D Stock

series ordinal

3

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20 October 2019

publication date

1 February 1996

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20 October 2019

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20 October 2019

volume

30

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20 October 2019

issue

1

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20 October 2019

page(s)

73-79

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Molecular pharmacology of V1a vasopressin receptors.

20 October 2019

cites work

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7 January 2021

No requirement of cyclic conformation of antagonists in binding to vasopressin receptors

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Design of potent and selective linear antagonists of vasopressor (V1-receptor) responses to vasopressin

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7 January 2021

Novel approach to the design of synthetic radioiodinated linear V1A receptor antagonists of vasopressin

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7 January 2021

Conformational and structural considerations in oxytocin-receptor binding and biological activity

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[1-beta-Mercapto-beta,beta-cyclopentamethylenepropionic acid),2-(O-methyl)tyrosine ]argine-vasopressin and [1-beta-mercapto-beta,beta-cyclopentamethylenepropionic acid)]argine-vasopressine, two highly potent antagonists of the vasopressor response t

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7 January 2021

A minor modification of residue 1 in potent vasopressin antagonists dramatically reduces agonist activity

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7 January 2021

Pharmacological characterization of linear analogues of vasopressin generated by the systematic substitution of positions 1 and 6 by L-amino acids

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7 January 2021

Potent and selective antagonists of the antidiuretic responses to arginine-vasopressin based on modifications of [1-(beta-mercapto-beta,beta-pentamethylenepropionic acid),2-D-isoleucine,4- valine]arginine-vasopressin at position 4

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7 January 2021

Fluorescent and biotinylated linear peptides as selective bifunctional ligands for the V1a vasopressin receptor.

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7 January 2021

A selective biotinylated probe for V1a vasopressin receptors

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

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Lack of V1 vasopressin receptors in rabbit hepatocytes

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7 January 2021

Hypothalamic regulatory hormones

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7 January 2021

Bombesin:potent effects on thermoregulation in the rat.

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Novel linear antagonists of the antidiuretic (V2) and vasopressor (V1) responses to vasopressin

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7 January 2021

2-O-alkyltyrosine derivatives of 1-deamino-arginine-vasopressin: highly specific and potent antidiuretic agonists

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7 January 2021

125I-labelled d(CH2)5[Tyr(Me)2,Thr4,Tyr-NH2(9)]OVT: a selective oxytocin receptor ligand

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7 January 2021

A radioiodinated linear vasopressin antagonist: a ligand with high affinity and specificity for V1a receptors

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7 January 2021

Design and synthesis of heterofunctional V1a-selective vasopressin receptor ligands with lysine at position 9

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7 January 2021

Characterization of the human liver vasopressin receptor. Profound differences between human and rat vasopressin-receptor-mediated responses suggest only a minor role for vasopressin in regulating human hepatic function

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7 January 2021

10.1016/S0143-4179(96)90058-X

Identifiers

DOI

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20 October 2019

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