Analysis of structural requirements for Ah receptor antagonist activity: ellipticines, flavones, and related compounds (Q71951714)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8986142%20AND%20SRC:MED&resulttype=core&format=json

22 October 2019

title

Analysis of structural requirements for Ah receptor antagonist activity: ellipticines, flavones, and related compounds (English)

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22 October 2019

author name string

T A Gasiewicz

1

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22 October 2019

A S Kende

2

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22 October 2019

G Rucci

3

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22 October 2019

B Whitney

4

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22 October 2019

J J Willey

5

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22 October 2019

language of work or name

English

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publication date

1 December 1996

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22 October 2019

published in

Biochemical Pharmacology

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22 October 2019

volume

52

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22 October 2019

issue

11

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22 October 2019

page(s)

1787-1803

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Mechanistic aspects of dioxin action

22 October 2019

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Mechanism of action of 2,3,7,8-tetrachlorodibenzo-p-dioxin antagonists: Characterization of 6-[125I]methyl-8-iodo-1, 3-dichlorodibenzofuran-Ah receptor complexes

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Binding characteristics of Ah receptors from rats and mice before and after separation from hepatic cytosols. 7-Hydroxyellipticine as a competitive antagonist of cytochrome P-450 induction

7 January 2021

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Inhibition of Ah (dioxin) receptor transformation by 9-hydroxy ellipticine. Involvement of protein kinase C?

7 January 2021

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Chelatable metal ions are not required for aryl hydrocarbon receptor transformation to a DNA binding form: phenanthrolines are possible competitive antagonists of 2,3,7,8-tetrachlorodibenzo-p-dioxin

7 January 2021

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Topoisomerase II-mediated DNA cleavage activity induced by ellipticines on the human tumor cell line N417.

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The examination and quantitation of tissue cytosolic receptors for 2,3,7,8-tetrachlorodibenzo-p-dioxin using hydroxylapatite

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

7 January 2021

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Dioxin-dependent activation of murine Cyp1a-1 gene transcription requires protein kinase C-dependent phosphorylation

7 January 2021

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Three-dimensional quantitative structure-activity relationships of dioxins and dioxin-like compounds: model validation and Ah receptor characterization

7 January 2021

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Identification of 3'-methoxy-4'-nitroflavone as a pure aryl hydrocarbon (Ah) receptor antagonist and evidence for more than one form of the nuclear Ah receptor in MCF-7 human breast cancer cells

7 January 2021

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7 January 2021

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Structure-activity relationships in the inhibitory effects of ellipticines on benzo(a)pyrene hydroxylase activity and 3-methylcholanthrene mutagenicity

7 January 2021

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7 January 2021

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10.1016/S0006-2952(96)00600-4

7 January 2021

Identifiers

DOI

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8986142%20AND%20SRC:MED&resulttype=core&format=json

22 October 2019

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