Potent active site-directed inhibition of steroid sulphatase by tricyclic coumarin-based sulphamates (Q73081554)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11033081%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

title

Potent active site-directed inhibition of steroid sulphatase by tricyclic coumarin-based sulphamates (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11033081%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

author name string

L L Woo

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11033081%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

A Purohit

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11033081%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

B Malini

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11033081%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

M J Reed

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11033081%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

B V Potter

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11033081%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

publication date

1 October 2000

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11033081%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

published in

Chemistry and Biology

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11033081%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

volume

7

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11033081%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

issue

10

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11033081%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

page(s)

773-791

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11033081%20AND%20SRC:MED&resulttype=core&format=json

New aromatase inhibitors: more selectivity, less toxicity, unfortunately, the same activity

1 November 2019

cites work

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Aromatase inhibitors--where are we now?

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

In situ estrogen production via the estrone sulfatase pathway in breast tumors: relative importance versus the aromatase pathway

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Estrogen productivity of endometrium and endometrial cancer tissue; influence of aromatase on proliferation of endometrial cancer cells

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

The plasma concentration of oestrone sulphate in postmenopausal women: lack of diurnal variation, effect of ovariectomy, age and weight

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Aromatase activity in normal breast and breast tumor tissues: in vivo and in vitro studies

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Estrogen sulfatase and estrogen sulfotransferase in human primary mammary carcinoma

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Estrone sulfate and sulfatase activity in human breast cancer and endometrial cancer

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Comparison of estrogen concentrations, estrone sulfatase and aromatase activities in normal, and in cancerous, human breast tissues

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Androstenedione and androst-5-ene-3 beta,17 beta-diol stimulate DMBA-induced rat mammary tumors--role of aromatase

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

DHEA and peripheral androgen and estrogen formation: intracinology

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

1 reference

7 January 2021

Dehydroepiandrosterone: Kinetics of Metabolism in Normal Men and Women*

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

The use of nonradiolabelled steroid infusions to investigate the origin of oestrone sulphate in postmenopausal women

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Hormones, peripherally activated prohormones and regulation of the Th1/Th2 balance.

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Reversal of scopolamine induced amnesia in rats by the steroid sulfatase inhibitor estrone-3-O-sulfamate.

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Enhanced plasma DHEAS, brain acetylcholine and memory mediated by steroid sulfatase inhibition

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Memory enhancement mediated by the steroid sulfatase inhibitor (p-O-sulfamoyl)-N-tetradecanoyl tyramine

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

The hydrolysis of oestrone sulphate and dehydroepiandrosterone sulphate by human steroid sulphatase expressed in transfected COS-1 cells

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Estrone sulfamates: potent inhibitors of estrone sulfatase with therapeutic potential

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Inactivation of steroid sulfatase by an active site-directed inhibitor, estrone-3-O-sulfamate

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

In vivo inhibition of oestrone sulphatase and dehydroepiandrosterone sulphatase by oestrone-3-O-sulphamate

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Steroidal and nonsteroidal sulfamates as potent inhibitors of steroid sulfatase

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Sulfamates of various estrogens are prodrugs with increased systemic and reduced hepatic estrogenicity at oral application

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Active site directed inhibition of estrone sulfatase by nonsteroidal coumarin sulfamates

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Estrone sulfatase: probing structural requirements for substrate and inhibitor recognition

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Synthesis and sulfatase inhibitory activities of non-steroidal estrone sulfatase inhibitors

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Development of potent non-estrogenic estrone sulfatase inhibitors

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Potent inhibition of steroid sulfatase activity by 3-O-sulfamate 17alpha-benzyl(or 4'-tert-butylbenzyl)estra-1,3,5(10)-trienes: combination of two substituents at positions C3 and c17alpha of estradiol

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Heteroatom-substituted analogues of the active-site directed inhibitor estra-1,3,5(10)-trien-17-one-3-sulphamate inhibit estrone sulphatase by a different mechanism

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Structure of a human lysosomal sulfatase

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Sulfatases, trapping of the sulfated enzyme intermediate by substituting the active site formylglycine

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Crystal structure of human arylsulfatase A: the aldehyde function and the metal ion at the active site suggest a novel mechanism for sulfate ester hydrolysis

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Amino acid residues forming the active site of arylsulfatase A. Role in catalytic activity and substrate binding

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

The development of A-ring modified analogues of oestrone-3-O-sulphamate as potent steroid sulphatase inhibitors with reduced oestrogenicity

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

A novel amino acid modification in sulfatases that is defective in multiple sulfatase deficiency

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Residues critical for formylglycine formation and/or catalytic activity of arylsulfatase A.

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

A cluster of sulfatase genes on Xp22.3: mutations in chondrodysplasia punctata (CDPX) and implications for warfarin embryopathy

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

Conversion of cysteine to formylglycine: a protein modification in the endoplasmic reticulum

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

The evolutionary conservation of a novel protein modification, the conversion of cysteine to serinesemialdehyde in arylsulfatase from Volvox carteri

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2800%2900023-5

7 January 2021

10.1016/S1074-5521(00)00023-5

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11033081%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

1 reference