Prediction of the intestinal absorption of endothelin receptor antagonists using three theoretical methods of increasing complexity (Q73163235)

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1 November 2019

title

Prediction of the intestinal absorption of endothelin receptor antagonists using three theoretical methods of increasing complexity (English)

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1 November 2019

author name string

P Stenberg

1

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1 November 2019

K Luthman

2

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1 November 2019

H Ellens

3

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1 November 2019

C P Lee

4

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1 November 2019

P L Smith

5

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1 November 2019

A Lago

6

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1 November 2019

J D Elliott

7

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1 November 2019

P Artursson

8

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publication date

1 October 1999

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1 November 2019

published in

Pharmaceutical Research

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1 November 2019

volume

16

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issue

10

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page(s)

1520-1526

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Theoretical calculation and prediction of Caco-2 cell permeability using MolSurf parametrization and PLS statistics

1 November 2019

cites work

1 reference

12 December 2020

Theoretical calculation and prediction of brain-blood partitioning of organic solutes using MolSurf parametrization and PLS statistics.

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A practitioner's perspective of the role of quantitative structure-activity analysis in medicinal chemistry

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Correlation of human jejunal permeability (in vivo) of drugs with experimentally and theoretically derived parameters. A multivariate data analysis approach

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12 December 2020

Membrane transport of drugs in different regions of the intestinal tract of the rat.

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12 December 2020

Intestinal drug absorption and metabolism in cell cultures: Caco-2 and beyond

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12 December 2020

Evaluation of dynamic polar molecular surface area as predictor of drug absorption: comparison with other computational and experimental predictors

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12 December 2020

Prediction of membrane permeability to peptides from calculated dynamic molecular surface properties

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12 December 2020

Nonpeptide endothelin receptor antagonists. VI: Pharmacological characterization of SB 217242, a potent and highly bioavailable endothelin receptor antagonist

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12 December 2020

Correlation of drug absorption with molecular surface properties

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12 December 2020

Prodrugs revisited: the "ad hoc" approach as a complement to ligand design

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12 December 2020

Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings

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12 December 2020

Automated absorption assessment using Caco-2 cells cultured on both sides of polycarbonate membranes

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12 December 2020

Caco-2 monolayers in experimental and theoretical predictions of drug transport

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12 December 2020

Physicochemical high throughput screening: parallel artificial membrane permeation assay in the description of passive absorption processes

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12 December 2020

Polar molecular surface properties predict the intestinal absorption of drugs in humans.

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12 December 2020

Identifiers

DOI

10.1023/A:1015092201811

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1 November 2019

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