A 6beta-(thiaheptanamide) derivative of estradiol as inhibitor of 17beta-hydroxysteroid dehydrogenase type 1 (Q74502716)

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11 November 2019

title

A 6beta-(thiaheptanamide) derivative of estradiol as inhibitor of 17beta-hydroxysteroid dehydrogenase type 1 (English)

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11 November 2019

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D Poirier

1

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11 November 2019

P Dionne

series ordinal

2

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11 November 2019

S Auger

series ordinal

3

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11 November 2019

publication date

1 January 1998

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The Journal of Steroid Biochemistry and Molecular Biology

11 November 2019

published in

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11 November 2019

volume

64

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11 November 2019

issue

1-2

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11 November 2019

page(s)

83-90

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11 November 2019

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Aromatase, 17 beta-hydroxysteroid dehydrogenase and intratissular sex hormone concentrations in cancerous and normal glandular breast tissue in postmenopausal women

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A comparison of the in vivo uptake and metabolism of 3H-oestrone and 3H-oestradiol by normal breast and breast tumour tissues in post-menopausal women

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The affinity alkylators, 11 alpha-bromoacetoxyprogesterone and estrone 3-bromoacetate, modify a common histidyl residue in the active site of human placental 17 beta,20 alpha-hydroxysteroid dehydrogenase

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Structure of the steroid-binding site of human placental estradiol-17β-dehydrogenase

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Alkylation of Estradiol 17beta-Dehydrogenase from Human Placenta with 3-Chloroacetylpyridine - Adenine Dinucleotide

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Affinity labeling of the cofactor-binding site of estradiol 17 beta-dehydrogenase of human placenta by 5'-p-fluorosulfonylbenzoyl adenosine

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7 January 2021

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7 January 2021

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Identifiers

DOI

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11 November 2019

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