Transport characteristics of peptidomimetics. Effect of the pyrrolinone bioisostere on transport across Caco-2 cell monolayers (Q74628282)

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12 November 2019

title

Transport characteristics of peptidomimetics. Effect of the pyrrolinone bioisostere on transport across Caco-2 cell monolayers (English)

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12 November 2019

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2

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12 November 2019

author name string

M Sudoh

1

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12 November 2019

W Yao

3

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12 November 2019

W Moser

4

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12 November 2019

A Yokoyama

5

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12 November 2019

A Pasternak

6

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12 November 2019

P A Sprengeler

7

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A B Smith

8

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R Hirschmann

9

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12 November 2019

R T Borchardt

10

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publication date

1 May 1998

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12 November 2019

number of pages

7

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inferred from page(s)

published in

Pharmaceutical Research

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12 November 2019

volume

15

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issue

5

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12 November 2019

page(s)

719-725

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Esterase-sensitive cyclic prodrugs of peptides: evaluation of an acyloxyalkoxy promoiety in a model hexapeptide

12 November 2019

cites work

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12 December 2020

Improvement of oral peptide bioavailability: Peptidomimetics and prodrug strategies

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12 December 2020

Epithelial transport of drugs in cell culture. I: A model for studying the passive diffusion of drugs over intestinal absorptive (Caco-2) cells

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12 December 2020

P-glycoprotein expression and function in circulating blood cells from normal volunteers.

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12 December 2020

Structure of complex of synthetic HIV-1 protease with a substrate-based inhibitor at 2.3 A resolution

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12 December 2020

Biochemistry of multidrug resistance mediated by the multidrug transporter

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12 December 2020

HIV protease: a novel chemotherapeutic target for AIDS.

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12 December 2020

An orally bioavailable pyrrolinone inhibitor of HIV-1 protease: computational analysis and X-ray crystal structure of the enzyme complex

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12 December 2020

Design and synthesis of peptidomimetic inhibitors of HIV-1 protease and renin. Evidence for improved transport

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12 December 2020

Antithrombotic agents: from RGD to peptide mimetics.

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12 December 2020

Expression of drug-metabolizing enzymes and P-170 glycoprotein in colorectal carcinoma and normal mucosa

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12 December 2020

Human serum alpha 1 acid glycoprotein reduces uptake, intracellular concentration, and antiviral activity of A-80987, an inhibitor of the human immunodeficiency virus type 1 protease.

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12 December 2020

Peptoids: a modular approach to drug discovery.

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12 December 2020

Predicting drug-membrane interactions by HPLC: structural requirements of chromatographic surfaces

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12 December 2020

L-735,524: an orally bioavailable human immunodeficiency virus type 1 protease inhibitor

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12 December 2020

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12 December 2020

Abnormal expression of a 170-kilodalton P-glycoprotein encoded by MDR1 gene, a metabolically active efflux pump, in CD4+ and CD8+ T cells from patients with human immunodeficiency virus type 1 infection

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12 December 2020

IAM chromatography: an in vitro screen for predicting drug membrane permeability

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12 December 2020

Discovery of a peptide-based renin inhibitor with oral bioavailability and efficacy

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12 December 2020

Evidence for a polarized efflux system for peptides in the apical membrane of Caco-2 cells

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12 December 2020

How structural features influence the biomembrane permeability of peptides

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12 December 2020

Identifiers

DOI

10.1023/A:1011966918959

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12 November 2019

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