Positive allosteric modulators of metabotropic glutamate 1 receptor: characterization, mechanism of action, and binding site (Q24555099)

2

V

Mutel

1 reference

19 October 2023

S Jolidon

3

S

Jolidon

1 reference

19 October 2023

J N Kew

4

J N

Kew

1 reference

19 October 2023

P Malherbe

5

P

Malherbe

1 reference

19 October 2023

E Vieira

6

E

Vieira

1 reference

19 October 2023

J Wichmann

7

J

Wichmann

1 reference

19 October 2023

J A Kemp

8

J A

Proceedings of the National Academy of Sciences of the United States of America

Kemp

1 reference

19 October 2023

language of work or name

English

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publication date

6 November 2001

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published in

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volume

98

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issue

23

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page(s)

13402-7

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cites work

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CPCCOEt, a noncompetitive metabotropic glutamate receptor 1 antagonist, inhibits receptor signaling without affecting glutamate binding

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Sequence and expression of a metabotropic glutamate receptor

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Pharmacological properties of native metabotropic glutamate receptors in freshly dissociated Golgi cells of the rat cerebellum

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The N-terminal domain of gamma-aminobutyric Acid(B) receptors is sufficient to specify agonist and antagonist binding.

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Changes in the carboxyl-terminal domain of metabotropic glutamate receptor 1 by alternative splicing generate receptors with differing agonist-independent activity.

30 May 2018

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Inhibition of calcium channels in rat CA3 pyramidal neurons by a metabotropic glutamate receptor

30 May 2018

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Characterization of [(3)H]Quisqualate binding to recombinant rat metabotropic glutamate 1a and 5a receptors and to rat and human brain sections

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28 November 2018

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Metabotropic glutamate receptors activate G-protein-coupled inwardly rectifying potassium channels in Xenopus oocytes.

28 November 2018

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Protein kinase C modulates glutamate receptor inhibition of Ca2+ channels and synaptic transmission.

28 November 2018

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Frequency detection and temporally dispersed synaptic signal association through a metabotropic glutamate receptor pathway

28 November 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/11606768

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

The non-competitive antagonists 2-methyl-6-(phenylethynyl)pyridine and 7-hydroxyiminocyclopropan[b]chromen-1a-carboxylic acid ethyl ester interact with overlapping binding pockets in the transmembrane region of group I metabotropic glutamate recepto

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/11606768

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Metabotropic glutamate receptors: electrophysiological properties and role in plasticity

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/11606768

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1073/PNAS.231358298

1 reference

release_baaxjpezufdtna24pfbqv3yxom

0 references

0 references

4793015

1 reference

1 reference

1 reference