Mechanisms of inhibition of HIV replication by non-nucleoside reverse transcriptase inhibitors (Q24652511)

Phenylethylthiazolylthiourea (PETT) non-nucleoside inhibitors of HIV-1 and HIV-2 reverse transcriptases. Structural and biochemical analyses

Europe PubMed Central

title

Mechanisms of inhibition of HIV replication by non-nucleoside reverse transcriptase inhibitors (English)

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Gilda Tachedjian

2

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Nicolas Sluis-Cremer

series ordinal

1

object named as

Nicolas Sluis-Cremer

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language of work or name

English

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publication date

June 2008

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published in

Virus Research

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volume

134

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page(s)

147-56

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issue

1-2

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cites work

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The activity of the protease of human immunodeficiency virus type 1 is initiated at the membrane of infected cells before the release of viral proteins and is required for release to occur with maximum efficiency.

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Proteolytic processing of an HIV-1 pol polyprotein precursor: insights into the mechanism of reverse transcriptase p66/p51 heterodimer formation

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Reverse transcriptase mutations 118I, 208Y, and 215Y cause HIV-1 hypersusceptibility to non-nucleoside reverse transcriptase inhibitors

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HIV-1 reverse transcriptase plus-strand initiation exhibits preferential sensitivity to non-nucleoside reverse transcriptase inhibitors in vitro

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Substrate-dependent inhibition or stimulation of HIV RNase H activity by non-nucleoside reverse transcriptase inhibitors (NNRTIs)

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The regulation of sequential processing of HIV-1 Gag by the viral protease

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Structural mapping of catalytic site with respect to alpha-subunit and noncatalytic site in yeast mitochondrial F1-ATPase using fluorescence resonance energy transfer

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PubMed

https://pubmed.ncbi.nlm.nih.gov/18372072

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12 December 2020

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Identifiers

DOI

10.1016/J.VIRUSRES.2008.01.002

1 reference

3352220

3352220

1 reference

1 reference

1 reference