Pharmacological profiles of a novel opioid receptor-like1 (ORL(1)) receptor antagonist, JTC-801 (Q24673352)

2

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Yasunori Suzuki

3

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Takao Ito

4

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Kazuo Aisaka

British Journal of Pharmacology

5

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language of work or name

English

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publication date

January 2002

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published in

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volume

135

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issue

2

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page(s)

323-32

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cites work

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Isolation and structure of the endogenous agonist of opioid receptor-like ORL1 receptor

7 April 2017

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4-Aminoquinolines: novel nociceptin antagonists with analgesic activity

7 April 2017

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[Phe1psi(CH2-NH)Gly2]nociceptin-(1-13)-NH2 is an agonist of the nociceptin (ORL1) receptor.

28 September 2017

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Isolation of a novel cDNA encoding a putative membrane receptor with high homology to the cloned mu, delta, and kappa opioid receptors.

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Molecular cloning and tissue distribution of a putative member of the rat opioid receptor gene family that is not a mu, delta or kappa opioid receptor type

28 September 2017

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Nociceptin (1 - 7) antagonizes nociceptin-induced hyperalgesia in mice

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Evidence that [Phe1 psi(CH2-NH)Gly2]nociceptin-(1-13)-NH2, a peripheral ORL-1 receptor antagonist, acts as an agonist in the rat spinal cord

30 May 2018

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30 May 2018

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A new selective antagonist of the nociceptin receptor.

30 May 2018

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Identification and characterization of an endogenous ligand for opioid receptor homologue ROR-C: its involvement in allodynic response to innocuous stimulus.

30 May 2018

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30 May 2018

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[Phe1psi(CH2-NH)Gly2]-nociceptin-(1-13)NH2, a proposed antagonist of the nociceptin receptor, is a potent and stable agonist in the rat spinal cord

30 May 2018

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Nociceptin (Orphanin FQ) abolishes gestational and ovarian sex steroid-induced antinociception and induces hyperalgesia

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Orphanin FQ: a neuropeptide that activates an opioidlike G protein-coupled receptor.

28 November 2018

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[Phe1psi(CH2-NH)Gly2]nociceptin-(1-13)-NH2 acts as an agonist of the orphanin FQ/nociceptin receptor in vivo

28 November 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/11815367

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Central administration of [Phe1psi(CH2-NH)Gly2]nociceptin(1-13)-NH2 and orphanin FQ/nociceptin (OFQ/N) produce similar cardiovascular and renal responses in conscious rats

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/11815367

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Intrathecal morphine in mice: a new technique

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/11815367