A surface on the androgen receptor that allosterically regulates coactivator binding (Q27648698)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242%20AND%20SRC:MED&resulttype=core&format=json

8 January 2020

title

A surface on the androgen receptor that allosterically regulates coactivator binding (English)

1 reference

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Correction for Estébanez-Perpiñá et al., A surface on the androgen receptor that allosterically regulates coactivator binding

8 January 2020

corrigendum / erratum

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author

Eva Estébanez-Perpiñá

1

1 reference

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8 January 2020

R. Kiplin Guy

10

1 reference

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8 January 2020

Leggy A Arnold

2

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Robert Fletterick

12

object named as

Robert J Fletterick

1 reference

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8 January 2020

11

Paul Webb

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8 January 2020

5

Ellena Mar

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8 January 2020

author name string

Phuong Nguyen

3

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8 January 2020

Edson Delgado Rodrigues

4

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8 January 2020

Raynard Bateman

6

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8 January 2020

Peter Pallai

7

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8 January 2020

Kevan M Shokat

8

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8 January 2020

John D Baxter

9

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8 January 2020

language of work or name

English

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publication date

2 October 2007

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Proceedings of the National Academy of Sciences of the United States of America

8 January 2020

published in

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8 January 2020

volume

104

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8 January 2020

page(s)

16074-16079

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8 January 2020

issue

41

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The molecular mechanisms of coactivator utilization in ligand-dependent transactivation by the androgen receptor

8 January 2020

cites work

1 reference

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7 April 2017

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7 April 2017

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7 April 2017

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Treatment of Postmenopausal Breast Cancer with Selective Estrogen Receptor Modulators (SERMs).

29 September 2017

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A second binding site for hydroxytamoxifen within the coactivator-binding groove of estrogen receptor beta

29 September 2017

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The expanding cosmos of nuclear receptor coactivators

29 September 2017

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Molecular regulation of androgen action in prostate cancer

29 September 2017

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Biology of progressive, castration-resistant prostate cancer: directed therapies targeting the androgen-receptor signaling axis

29 September 2017

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Development of peptide antagonists for the androgen receptor using combinatorial peptide phage display

29 September 2017

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Ligand control of coregulator recruitment to nuclear receptors

29 September 2017

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Signature of the oligomeric behaviour of nuclear receptors at the sequence and structural level

29 September 2017

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Finding specificity within a conserved interaction site

29 September 2017

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Modulation of protein-protein interactions with small organic molecules

29 September 2017

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The development of COX2 inhibitors

29 September 2017

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Androgen receptor mutations and androgen insensitivity

29 September 2017

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29 September 2017

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The NH(2)-terminal and carboxyl-terminal interaction in the human androgen receptor

29 September 2017

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Structure-based design and synthesis of a thyroid hormone receptor (TR) antagonist.

29 September 2017

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Mutations at the boundary of the hinge and ligand binding domain of the androgen receptor confer increased transactivation function

29 September 2017

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Discovering novel ligands for macromolecules using X-ray crystallographic screening

29 September 2017

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Human androgen receptor mutation disrupts ternary interactions between ligand, receptor domains, and the coactivator TIF2 (transcription intermediary factor 2).

29 September 2017

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Crossref

https://api.crossref.org/works/10.1073%2FPNAS.0708036104

Novel molecular defects in the androgen receptor gene of Mexican patients with androgen insensitivity

21 January 2018

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Crossref

https://api.crossref.org/works/10.1073%2FPNAS.0708036104

Dihydrotestosterone (DHT) modulates the ability of NSAIDs to induce apoptosis of prostate cancer cells

21 January 2018

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Functional analysis of 44 mutant androgen receptors from human prostate cancer.

21 January 2018

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Drug discovery at signaling interfaces

27 November 2018

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12 December 2020

Structural basis for androgen receptor interdomain and coactivator interactions suggests a transition in nuclear receptor activation function dominance

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12 December 2020

A high-throughput screening method to identify small molecule inhibitors of thyroid hormone receptor coactivator binding

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12 December 2020

Collocation of androgen receptor gene mutations in prostate cancer

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12 December 2020

Identifiers

DOI

10.1073/PNAS.0708036104

2 references

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242%20AND%20SRC:MED&resulttype=core&format=json

8 January 2020

ADS bibcode

2007PNAS..10416074E

0 references

1 reference

2 references

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242%20AND%20SRC:MED&resulttype=core&format=json

8 January 2020

2 references