6-Ethynylthieno[3,2-d]- and 6-ethynylthieno[2,3-d]pyrimidin-4-anilines as tunable covalent modifiers of ErbB kinases (Q27649889)

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3 January 2020

title

6-Ethynylthieno[3,2-d]- and 6-ethynylthieno[2,3-d]pyrimidin-4-anilines as tunable covalent modifiers of ErbB kinases (English)

1 reference

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Correction for Wood , 6-Ethynylthieno[3,2-d]- and 6-ethynylthieno[2,3-d]pyrimidin-4-anilines as tunable covalent modifiers of ErbB kinases

3 January 2020

corrigendum / erratum

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author

Dana E Vanderwall

21

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3 January 2020

author name string

Edgar R Wood

1

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3 January 2020

Lisa M Shewchuk

2

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3 January 2020

Byron Ellis

3

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3 January 2020

Perry Brignola

4

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3 January 2020

Ronald L Brashear

5

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3 January 2020

Thomas R Caferro

6

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3 January 2020

Scott H Dickerson

7

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Hamilton D Dickson

8

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Kelly H Donaldson

9

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Michael Gaul

10

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Robert J Griffin

11

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Anne M Hassell

12

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Barry Keith

13

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3 January 2020

Robert Mullin

14

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Kimberly G Petrov

15

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Michael J Reno

16

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David W Rusnak

17

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Sarva M Tadepalli

18

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John C Ulrich

19

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Craig D Wagner

20

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Alex G Waterson

22

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Jon D Williams

23

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Wendy L White

24

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David E Uehling

25

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language of work or name

English

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publication date

19 February 2008

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Proceedings of the National Academy of Sciences of the United States of America

3 January 2020

number of pages

6

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based on heuristic

inferred from page(s)

published in

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volume

105

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3 January 2020

issue

8

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3 January 2020

page(s)

2773-2778

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Structures of Lung Cancer-Derived EGFR Mutants and Inhibitor Complexes: Mechanism of Activation and Insights into Differential Inhibitor Sensitivity

3 January 2020

cites work

1 reference

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Structure-guided development of affinity probes for tyrosine kinases using chemical genetics

20 March 2017

1 reference

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An allosteric mechanism for activation of the kinase domain of epidermal growth factor receptor

20 March 2017

1 reference

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Structure of the epidermal growth factor receptor kinase domain alone and in complex with a 4-anilinoquinazoline inhibitor

20 March 2017

1 reference

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The characterization of novel, dual ErbB-2/EGFR, tyrosine kinase inhibitors: potential therapy for cancer

20 March 2017

1 reference

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A unique structure for epidermal growth factor receptor bound to GW572016 (Lapatinib): relationships among protein conformation, inhibitor off-rate, and receptor activity in tumor cells

20 March 2017

1 reference

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Specific, irreversible inactivation of the epidermal growth factor receptor and erbB2, by a new class of tyrosine kinase inhibitor

20 March 2017

1 reference

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Protein open-access liquid chromatography/mass spectrometry

20 March 2017

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Antitumor activity of HKI-272, an orally active, irreversible inhibitor of the HER-2 tyrosine kinase

29 September 2017

1 reference

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The effects of the novel, reversible epidermal growth factor receptor/ErbB-2 tyrosine kinase inhibitor, GW2016, on the growth of human normal and tumor-derived cell lines in vitro and in vivo.

29 September 2017

1 reference

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Small molecule inhibitors of the class 1 receptor tyrosine kinase family

29 September 2017

1 reference

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Comparison of the biochemical and kinetic properties of the type 1 receptor tyrosine kinase intracellular domains. Demonstration of differential sensitivity to kinase inhibitors

29 September 2017

1 reference

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Synthesis and structure-activity relationships of 6,7-disubstituted 4-anilinoquinoline-3-carbonitriles. The design of an orally active, irreversible inhibitor of the tyrosine kinase activity of the epidermal growth factor receptor (EGFR) and the hum

29 September 2017

1 reference

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27 November 2018

Identifiers

DOI

10.1073/PNAS.0708281105

1 reference

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3 January 2020

0 references

1 reference

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3 January 2020

PubMed publication ID

18287036

1 reference