6-Azido-7-nitro-1,4-dihydroquinoxaline-2,3-dione (ANQX) Forms an Irreversible Bond To the Active Site of the GluR2 AMPA Receptor † (Q27651830)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18754610%20AND%20SRC:MED&resulttype=core&format=json

13 January 2020

title

6-Azido-7-nitro-1,4-dihydroquinoxaline-2,3-dione (ANQX) forms an irreversible bond to the active site of the GluR2 AMPA receptor (English)

1 reference

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13 January 2020

0 references

Eva Estébanez-Perpiñá

2

1 reference

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13 January 2020

7

Robert J Fletterick

1 reference

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13 January 2020

author name string

Leslie A Cruz

1

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13 January 2020

Sam Pfaff

3

1 reference

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13 January 2020

Sabine Borngraeber

4

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13 January 2020

Ning Bao

5

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13 January 2020

Justin Blethrow

6

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13 January 2020

Pamela M England

8

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13 January 2020

language of work or name

English

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publication date

1 September 2008

1 reference

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Journal of Medicinal Chemistry

13 January 2020

published in

1 reference

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13 January 2020

volume

51

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13 January 2020

issue

18

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13 January 2020

page(s)

5856-5860

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TARP auxiliary subunits switch AMPA receptor antagonists into partial agonists

13 January 2020

cites work

1 reference

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Structural basis for partial agonist action at ionotropic glutamate receptors

20 March 2017

1 reference

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Probing the function, conformational plasticity, and dimer-dimer contacts of the GluR2 ligand-binding core: studies of 5-substituted willardiines and GluR2 S1S2 in the crystal

20 March 2017

1 reference

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Structural basis for AMPA receptor activation and ligand selectivity: crystal structures of five agonist complexes with the GluR2 ligand-binding core

20 March 2017

1 reference

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Mechanism of glutamate receptor desensitization

20 March 2017

1 reference

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Mechanisms for activation and antagonism of an AMPA-sensitive glutamate receptor: crystal structures of the GluR2 ligand binding core

20 March 2017

1 reference

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Structure of a glutamate-receptor ligand-binding core in complex with kainate

20 March 2017

1 reference

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A synaptic model of memory: long-term potentiation in the hippocampus

20 March 2017

1 reference

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The glutamate receptor ion channels

20 March 2017

1 reference

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Mechanism of positive allosteric modulators acting on AMPA receptors

20 March 2017

1 reference

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Distinct molecular mechanisms and divergent endocytotic pathways of AMPA receptor internalization

20 March 2017

1 reference

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Receptor trafficking and synaptic plasticity

20 March 2017

1 reference

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AMPA receptor trafficking and synaptic plasticity

7 April 2017

1 reference

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AMPA Receptor Trafficking at Excitatory Synapses

7 April 2017

1 reference

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Cloned glutamate receptors

7 April 2017

1 reference

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Photoinactivation of native AMPA receptors reveals their real-time trafficking

7 April 2017

1 reference

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Glutamate receptor ion channels

29 September 2017

1 reference

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The molecular pharmacology and cell biology of alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptors

29 September 2017

1 reference

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Structure and function of AMPA receptors

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2945402

Regulation of AMPA receptors during synaptic plasticity

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2945402

AMPA receptor antagonists

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2945402

Rapid photoinactivation of native AMPA receptors on live cells using ANQX.

29 September 2017

1 reference

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Photochemically knocking out glutamate receptors in vivo

27 November 2018

1 reference

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27 November 2018

Identifiers

DOI

10.1021/JM701517B

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18754610%20AND%20SRC:MED&resulttype=core&format=json

13 January 2020

1 reference

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13 January 2020

PubMed publication ID

18754610

1 reference