Discovery of a Novel Class of Covalent Inhibitor for Aldehyde Dehydrogenases (Q27675184)

10

Daria Mochly-Rosen

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Samantha Perez-Miller

Samantha Perez-Miller

5

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Ann Kimble-Hill

Ann Kimble-Hill

3

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May Khanna

May Khanna

1

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author name string

Che-Hong Chen

2

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Bibek Parajuli

4

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Sulochanadevi Baskaran

6

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Jeewon Kim

7

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Karl Dria

8

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Thomas D Hurley

Journal of Biological Chemistry

11

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language of work or name

English

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publication date

16 December 2011

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published in

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volume

286

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issue

50

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page(s)

43486-94

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cites work

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Suppression of heavy drinking and alcohol seeking by a selective ALDH-2 inhibitor

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Interaction of human aldehyde dehydrogenase with aromatic substrates and ligands

21 January 2018

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Identification of early intermediates of caspase activation using selective inhibitors and activity-based probes

21 January 2018

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Purification of liver aldehyde dehydrogenase by p-hydroxyacetophenone-sepharose affinity matrix and the coelution of chloramphenicol acetyl transferase from the same matrix with recombinantly expressed aldehyde dehydrogenase

21 January 2018

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Role of aldehyde dehydrogenase in cyclophosphamide-resistant L1210 leukemia

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12 December 2020

Selective carboxymethylation of cysteine-174 of the beta 2 beta 2 and beta 1 beta 1 human liver alcohol dehydrogenase isoenzymes by iodoacetate

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12 December 2020

Detoxification of cyclophosphamide by human aldehyde dehydrogenase isozymes

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12 December 2020

Involvement of glutamate 399 and lysine 192 in the mechanism of human liver mitochondrial aldehyde dehydrogenase

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12 December 2020

Cellular levels of class 1 and class 3 aldehyde dehydrogenases and certain other drug-metabolizing enzymes in human breast malignancies

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12 December 2020

A novel polymorphism (-357 G/A) of the ALDH2 gene: linkage disequilibrium and an association with alcoholism

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12 December 2020

Identifiers

DOI

10.1074/JBC.M111.293597

1 reference

1 reference

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PubMed publication ID

22021038

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