Discovery of a Novel Class of Orally Active Trypanocidal N -Myristoyltransferase Inhibitors (Q27676019)

David A Robinson

4

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Ruth Brenk

Ruth Brenk

15

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Paul G. Wyatt

Paul G Wyatt

19

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Ian H. Gilbert

Ian H Gilbert

20

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Alan Fairlamb

Alan H Fairlamb

16

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Laste Stojanovski

12

Laste Stojanovski

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Kevin D Read

18

Kevin D Read

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Michael J. Ferguson

17

Michael A J Ferguson

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Daniel Spinks

9

Daniel Spinks

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Irene Hallyburton

6

Irene Hallyburton

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Neil Richard Norcross

8

Neil R Norcross

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Suzanne Norval

11

Suzanne Norval

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Julie A Frearson

14

Julie A Frearson

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Leah S Torrie

13

Leah S Torrie

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Tracy Bayliss

10

Tracy Bayliss

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author name string

Laura A T Cleghorn

2

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Stuart P McElroy

3

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Victoria C Smith

5

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Justin R Harrison

Journal of Medicinal Chemistry

7

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language of work or name

English

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publication date

12 January 2012

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published in

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volume

55

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issue

1

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page(s)

140-52

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cites work

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ARL1 has an essential role in Trypanosoma brucei

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PubMed

https://pubmed.ncbi.nlm.nih.gov/22148754

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Processing of X-ray diffraction data collected in oscillation mode

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22148754

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Scanning alanine mutagenesis and de-peptidization of a Candida albicans myristoyl-CoA:protein N-myristoyltransferase octapeptide substrate reveals three elements critical for molecular recognition

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PubMed

https://pubmed.ncbi.nlm.nih.gov/22148754

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/JM201091T

1 reference

1975182

1975182

1 reference

1 reference

1 reference