Structure and dynamics of the M3 muscarinic acetylcholine receptor (Q27677433)

Albert C Pan

3

0 references

William I Weis

William I Weis

12

0 references

Brian Kobilka

14

Brian K Kobilka

0 references

Pil Seok Chae

9

Pil Seok Chae

0 references

Ron Ofer Dror

10

Ron O Dror

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author name string

Andrew C Kruse

1

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Jianxin Hu

2

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Daniel H Arlow

4

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Daniel M Rosenbaum

5

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Hillary F Green

7

0 references

Tong Liu

8

0 references

David E Shaw

11

0 references

Jürgen Wess

Structure of the human M2 muscarinic acetylcholine receptor bound to an antagonist

13

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language of work or name

English

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publication date

22 February 2012

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published in

Nature

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volume

482

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issue

7386

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page(s)

552-6

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cites work

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Mapping of single amino acid residues required for selective activation of Gq/11 by the m3 muscarinic acetylcholine receptor

20 March 2017

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The M3-muscarinic receptor regulates learning and memory in a receptor phosphorylation/arrestin-dependent manner

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The constitutive activity of the human muscarinic M3 receptor unmasks differences in the pharmacology of anticholinergics

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Neuronal M3 muscarinic acetylcholine receptors are essential for somatotroph proliferation and normal somatic growth

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Mutagenic mapping suggests a novel binding mode for selective agonists of M1 muscarinic acetylcholine receptors

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Mice lacking the M3 muscarinic acetylcholine receptor are hypophagic and lean.

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2 June 2018

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2 June 2018

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Pronounced conformational changes following agonist activation of the M(3) muscarinic acetylcholine receptor

27 November 2018

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Conformational changes that occur during M3 muscarinic acetylcholine receptor activation probed by the use of an in situ disulfide cross-linking strategy

27 November 2018

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Multiple residues in the second extracellular loop are critical for M3 muscarinic acetylcholine receptor activation

27 November 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/22358844

12 December 2020

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1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22358844

12 December 2020

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Crossref

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Identifiers

DOI

10.1038/NATURE10867

1 reference

Dimensions Publication ID

877443

1002311039

0 references

877443

1 reference

1 reference

1 reference