Structure-guided Development of Specific Pyruvate Dehydrogenase Kinase Inhibitors Targeting the ATP-binding Pocket (Q27680986)

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3 March 2020

title

Structure-guided development of specific pyruvate dehydrogenase kinase inhibitors targeting the ATP-binding pocket (English)

1 reference

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3 March 2020

0 references

1 reference

2

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3 March 2020

Cheng-Yang Wu

4

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Ingrid Wernstedt Asterholm

3 March 2020

6

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3 March 2020

Kyle Owens

8

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3 March 2020

Richard M Wynn

12

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3 March 2020

9

Philipp E Scherer

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3 March 2020

author name string

Shih-Chia Tso

1

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3 March 2020

Wen-Jun Gui

3

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3 March 2020

Jacinta L Chuang

5

1 reference

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3 March 2020

Lorraine K Morlock

7

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3 March 2020

Noelle S Williams

10

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3 March 2020

Uttam K Tambar

11

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3 March 2020

David T Chuang

13

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3 March 2020

language of work or name

English

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publication date

19 December 2013

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Journal of Biological Chemistry

3 March 2020

number of pages

12

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based on heuristic

inferred from page(s)

published in

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3 March 2020

volume

289

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3 March 2020

issue

7

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3 March 2020

page(s)

4432-4443

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3 March 2020

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Regulatory roles of the N-terminal domain based on crystal structures of human pyruvate dehydrogenase kinase 2 containing physiological and synthetic ligands

20 March 2017

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20 March 2017

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20 March 2017

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21 January 2018

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21 January 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/24356970

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Secondary amides of (R)-3,3,3-trifluoro-2-hydroxy-2-methylpropionic acid as inhibitors of pyruvate dehydrogenase kinase

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24356970

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1074/JBC.M113.533885

2 references

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3 March 2020

1 reference

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3 March 2020

2 references

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