Mapping the rho1 GABA(C) receptor agonist binding pocket. Constructing a complete model (Q28293890)

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Stanislav O Zakharkin

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Delores Davis

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David S Weiss

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Yongchang Chang

Journal of Biological Chemistry

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language of work or name

English

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publication date

14 January 2005

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published in

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volume

280

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issue

2

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page(s)

1535-42

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cites work

GABAC receptors: relatively simple transmitter-gated ion channels?

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GABAA receptor needs two homologous domains of the beta-subunit for activation by GABA but not by pentobarbital

21 January 2018

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GABA(A) receptor beta 2 Tyr97 and Leu99 line the GABA-binding site. Insights into mechanisms of agonist and antagonist actions

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The GABAA receptor alpha 1 subunit Pro174-Asp191 segment is involved in GABA binding and channel gating

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Nicotinic receptors at the amino acid level

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Crystal structure of an ACh-binding protein reveals the ligand-binding domain of nicotinic receptors

21 January 2018

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Identification of a tyrosine in the agonist binding site of the homomeric rho1 gamma-aminobutyric acid (GABA) receptor that, when mutated, produces spontaneous opening

21 January 2018

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Acetylcholine receptor channel structure probed in cysteine-substitution mutants.

21 January 2018

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Identification of channel-lining residues in the M2 membrane-spanning segment of the GABA(A) receptor alpha1 subunit

21 January 2018

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The location of the gate in the acetylcholine receptor channel

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Different residues in the GABA(A) receptor alpha 1T60-alpha 1K70 region mediate GABA and SR-95531 actions

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Mapping the agonist binding site of the nicotinic acetylcholine receptor by cysteine scanning mutagenesis: antagonist footprint and secondary structure prediction

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Mapping the agonist binding site of the nicotinic acetylcholine receptor. Orientation requirements for activation by covalent agonist

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Channel opening locks agonist onto the GABAC receptor

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SWISS-MODEL: An automated protein homology-modeling server

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Crystallography & NMR System: A New Software Suite for Macromolecular Structure Determination

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Site-specific fluorescence reveals distinct structural changes with GABA receptor activation and antagonism

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Binding, gating, affinity and efficacy: the interpretation of structure-activity relationships for agonists and of the effects of mutating receptors

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Insights into the activation mechanism of rho1 GABA receptors obtained by coexpression of wild type and activation-impaired subunits.

21 January 2018

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Allosteric activation mechanism of the alpha 1 beta 2 gamma 2 gamma-aminobutyric acid type A receptor revealed by mutation of the conserved M2 leucine

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Agonist-induced closure of constitutively open gamma-aminobutyric acid channels with mutated M2 domains

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release_vdiqfdury5fn3ciqox3uvtlegy

21 January 2018

Identifiers

DOI

10.1074/JBC.M409908200

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Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/vdiqfdury5fn3ciqox3uvtlegy