Discovery and in vivo evaluation of new melanocortin-4 receptor-selective peptides. (Q30909790)

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2 November 2019

title

Discovery and in vivo evaluation of new melanocortin-4 receptor-selective peptides (English)

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2 November 2019

9

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2 November 2019

10

Roger A H Adan

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2 November 2019

author name string

Wouter A J Nijenhuis

1

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2 November 2019

John A W Kruijtzer

2

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2 November 2019

Nienke Wanders

3

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2 November 2019

Dorien H Vrinten

4

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2 November 2019

Keith M Garner

5

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2 November 2019

Wim M M Schaaper

6

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2 November 2019

Rob H Meloen

7

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2 November 2019

Willem Hendrik Gispen

8

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2 November 2019

publication date

1 February 2003

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2 November 2019

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2 November 2019

volume

24

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2 November 2019

issue

2

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2 November 2019

page(s)

271-280

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Characterization of melanocortin receptor ligands on cloned brain melanocortin receptors and on grooming behavior in the rat

2 November 2019

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Analogs of MTII, lactam derivatives of alpha-melanotropin, modified at the N-terminus, and their selectivity at human melanocortin receptors 3, 4, and 5

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Selective, high affinity peptide antagonists of alpha-melanotropin action at human melanocortin receptor 4: their synthesis and biological evaluation in vitro

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Potent and selective peptide agonists of alpha-melanotropin action at human melanocortin receptor 4: their synthesis and biological evaluation in vitro.

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Structure-function studies on the cyclic peptide MT-II, lactam derivative of alpha-melanotropin

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Inactivation of the mouse melanocortin-3 receptor results in increased fat mass and reduced lean body mass

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Characterization of melanocortin NDP-MSH agonist peptide fragments at the mouse central and peripheral melanocortin receptors

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Structure activity studies of the melanocortin antagonist SHU9119 modified at the 6, 7, 8, and 9 positions

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Biological and conformational examination of stereochemical modifications using the template melanotropin peptide, Ac-Nle-c[Asp-His-Phe-Arg-Trp-Ala-Lys]-NH2, on human melanocortin receptors

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Cyclic lactam alpha-melanotropin analogues of Ac-Nle4-cyclo[Asp5, D-Phe7,Lys10] alpha-melanocyte-stimulating hormone-(4-10)-NH2 with bulky aromatic amino acids at position 7 show high antagonist potency and selectivity at specific melanocortin recep

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alpha-Melanotropin: the minimal active sequence in the frog skin bioassay

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