Identification of small-molecule antagonists that inhibit an activator: coactivator interaction (Q31134749)

23 September 2017

Identification of small-molecule antagonists that inhibit an activator: coactivator interaction (English)

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23 September 2017

8

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23 September 2017

Tsaffrir Zor

7

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Bernhard Mayr

object named as

Bernhard Mayr

3

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author name string

Jennifer L Best

1

1 reference

23 September 2017

Carlos A Amezcua

2

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23 September 2017

Lawrence Flechner

4

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23 September 2017

Christopher M Murawsky

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23 September 2017

Beverly Emerson

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23 September 2017

Marc Montminy

9

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23 September 2017

language of work or name

English

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publication date

7 December 2004

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Proceedings of the National Academy of Sciences of the United States of America

23 September 2017

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23 September 2017

101

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23 September 2017

51

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23 September 2017

17622-17627

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describes a project that uses

23 September 2017

ImageQuant

1 reference

11 June 2022

https://www.ebi.ac.uk/europepmc/webservices/rest/PMC539725/fullTextXML

based on heuristic

inferred from PubMed Central ID database lookup

cites work

NMR View: A computer program for the visualization and analysis of NMR data

1 reference

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In vivo activation of the p53 pathway by small-molecule antagonists of MDM2

21 June 2018

1 reference

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TORCs: transducers of regulated CREB activity

21 June 2018

1 reference

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Identification of a family of cAMP response element-binding protein coactivators by genome-scale functional analysis in mammalian cells

21 June 2018

1 reference

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Structure and interactions of PAS kinase N-terminal PAS domain: model for intramolecular kinase regulation

21 June 2018

1 reference

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Cooperativity in transcription factor binding to the coactivator CREB-binding protein (CBP). The mixed lineage leukemia protein (MLL) activation domain binds to an allosteric site on the KIX domain

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=539725

Roles of phosphorylation and helix propensity in the binding of the KIX domain of CREB-binding protein by constitutive (c-Myb) and inducible (CREB) activators

21 June 2018

1 reference

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A transcriptional switch mediated by cofactor methylation

21 June 2018

1 reference

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CREB regulates hepatic gluconeogenesis through the coactivator PGC-1

21 June 2018

1 reference

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Control of hepatic gluconeogenesis through the transcriptional coactivator PGC-1

21 June 2018

1 reference

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Distinct effects of cAMP and mitogenic signals on CREB-binding protein recruitment impart specificity to target gene activation via CREB.

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=539725

MLL and CREB bind cooperatively to the nuclear coactivator CREB-binding protein

21 June 2018

1 reference

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HATs off: selective synthetic inhibitors of the histone acetyltransferases p300 and PCAF.

21 June 2018

1 reference

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Characterization of a CREB gain-of-function mutant with constitutive transcriptional activity in vivo

21 June 2018

1 reference

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Role of secondary structure in discrimination between constitutive and inducible activators

21 June 2018

1 reference

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Analysis of an activator:coactivator complex reveals an essential role for secondary structure in transcriptional activation

21 June 2018

1 reference

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Phosphorylation of NF-kappa B p65 by PKA stimulates transcriptional activity by promoting a novel bivalent interaction with the coactivator CBP/p300

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=539725

Solution Structure of the KIX Domain of CBP Bound to the Transactivation Domain of CREB: A Model for Activator:Coactivator Interactions

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=539725

Transcriptional activation by recruitment

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=539725

Discovering high-affinity ligands for proteins: SAR by NMR

21 June 2018

1 reference

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Phosphorylation of CREB at Ser-133 induces complex formation with CREB-binding protein via a direct mechanism

21 June 2018

1 reference

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NMRPipe: a multidimensional spectral processing system based on UNIX pipes

21 June 2018

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Structural analyses of CREB-CBP transcriptional activator-coactivator complexes by NMR spectroscopy: implications for mapping the boundaries of structural domains

21 June 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0406374101

Solution structure of the KIX domain of CBP bound to the transactivation domain of c-Myb

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0406374101

Contribution to stability and folding of a buried polar residue at the CARM1 methylation site of the KIX domain of CBP.

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0406374101

Transcriptional regulation by p53 through intrinsic DNA/chromatin binding and site-directed cofactor recruitment.

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0406374101

Genome-wide analysis of CREB target genes reveals a core promoter requirement for cAMP responsiveness

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0406374101

Structurally distinct modes of recognition of the KIX domain of CBP by Jun and CREB.

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0406374101

Structure and Interactions of PAS Kinase N-Terminal PAS Domain

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0406374101

21 January 2018

Identifiers

DOI

10.1073/PNAS.0406374101

1 reference

23 September 2017

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23 September 2017

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