Design and synthesis of new bicyclic diketopiperazines as scaffolds for receptor probes of structurally diverse functionality. (Q31172630)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15889186%20AND%20SRC:MED&resulttype=core&format=json

11 January 2020

title

Design and synthesis of new bicyclic diketopiperazines as scaffolds for receptor probes of structurally diverse functionality (English)

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11 January 2020

4

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11 January 2020

Kenneth A. Jacobson

series ordinal

5

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11 January 2020

Craig J Thomas

3

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ORCID Public Data File 2021

author name string

Pedro Besada

series ordinal

1

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11 January 2020

Liaman Mamedova

series ordinal

2

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11 January 2020

publication date

21 April 2005

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Organic and Biomolecular Chemistry

11 January 2020

published in

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11 January 2020

volume

3

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11 January 2020

issue

10

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11 January 2020

page(s)

2016-2025

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Discovery of an inhibitor of a transcription factor using small molecule microarrays and diversity-oriented synthesis

11 January 2020

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28 July 2018

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Synthesis and activity of a new generation of ruthenium-based olefin metathesis catalysts coordinated with 1,3-dimesityl-4,5-dihydroimidazol-2-ylidene ligands

28 July 2018

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A G protein-coupled receptor for UDP-glucose

28 July 2018

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Structure-activity relationships of bisphosphate nucleotide derivatives as P2Y1 receptor antagonists and partial agonists.

28 July 2018

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Rational design and combinatorial evaluation of enzyme inhibitor scaffolds: identification of novel inhibitors of matrix metalloproteinases

28 July 2018

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Identification of potent P2Y-purinoceptor agonists that are derivatives of adenosine 5'-monophosphate

28 July 2018

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Identification of potent, selective P2Y-purinoceptor agonists: structure-activity relationships for 2-thioether derivatives of adenosine 5'-triphosphate

28 July 2018

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A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

28 July 2018

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Architecture of P2Y nucleotide receptors: structural comparison based on sequence analysis, mutagenesis, and homology modeling.

28 July 2018

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Nucleotide analogues containing 2-oxa-bicyclo[2.2.1]heptane and l-alpha-threofuranosyl ring systems: interactions with P2Y receptors

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31 October 2018

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Design, synthesis, and conformational analysis of eight-membered cyclic peptidomimetics prepared using ring closing metathesis

31 October 2018

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A general approach toward the synthesis of C-nucleoside pyrazolo[1,5-a]-1,3,5-triazines and their 3',5'-bisphosphate C-nucleotide analogues as the first reported in vivo stable P2Y(1)-receptor antagonists

31 October 2018

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Acyclic and cyclopropyl analogues of adenosine bisphosphate antagonists of the P2Y1 receptor: structure-activity relationships and receptor docking

31 October 2018

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Identification of the platelet ADP receptor targeted by antithrombotic drugs

31 October 2018

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31 October 2018

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31 October 2018

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12 December 2020

TAN-1496 A, C and E, diketopiperazine antibiotics with inhibitory activity against mammalian DNA topoisomerase I

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12 December 2020

2-thioether 5'-O-(1-thiotriphosphate)adenosine derivatives as new insulin secretagogues acting through P2Y-Receptors

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12 December 2020

Solid-phase synthesis and structural characterization of highly substituted hydroxyproline-based 2,5-diketopiperazines

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Recent developments in olefin cross-metathesis

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12 December 2020

Identifiers

DOI

10.1039/B416349D

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15889186%20AND%20SRC:MED&resulttype=core&format=json

11 January 2020

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11 January 2020

PubMed publication ID

15889186

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