Structure and dynamics of the GABA binding pocket: A narrowing cleft that constricts during activation. (Q31813374)

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3 November 2019

title

Structure and dynamics of the GABA binding pocket: A narrowing cleft that constricts during activation (English)

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3 November 2019

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D A Wagner

1

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3 November 2019

C Czajkowski

series ordinal

2

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3 November 2019

language of work or name

English

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publication date

1 January 2001

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3 November 2019

published in

Journal of Neuroscience

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3 November 2019

volume

21

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3 November 2019

issue

1

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3 November 2019

page(s)

67-74

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Decreased agonist sensitivity of human GABA(A) receptors by an amino acid variant, isoleucine to valine, in the alpha1 subunit

3 November 2019

cites work

1 reference

12 December 2020

Distinct agonist- and antagonist-binding sites on the glycine receptor

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Mapping the agonist binding site of the GABAA receptor: evidence for a beta-strand.

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Activation and block of recombinant GABA(A) receptors by pentobarbitone: a single-channel study

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Agonist-induced changes in substituted cysteine accessibility reveal dynamic extracellular structure of M3-M4 loop of glutamate receptor GluR6.

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Binding, gating, affinity and efficacy: the interpretation of structure-activity relationships for agonists and of the effects of mutating receptors

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Amino acids of the Torpedo marmorata acetylcholine receptor alpha subunit labeled by a photoaffinity ligand for the acetylcholine binding site

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Reactivity of small thiolate anions and cysteine-25 in papain toward methyl methanethiosulfonate

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Improved secondary structure predictions for a nicotinic receptor subunit: incorporation of solvent accessibility and experimental data into a two-dimensional representation

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12 December 2020

Relationships between inhibition constants and fractional inhibition in enzyme-catalyzed reactions with different numbers of reactants, different reaction mechanisms, and different types and mechanisms of inhibition.

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GABAA receptor needs two homologous domains of the beta-subunit for activation by GABA but not by pentobarbital.

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Point mutations affecting antagonist affinity and agonist dependent gating of GABAA receptor channels.

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Bicuculline and gabazine are allosteric inhibitors of channel opening of the GABAA receptor

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Evolutionary history of the ligand-gated ion-channel superfamily of receptors

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Propofol increases agonist efficacy at the GABA(A) receptor.

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The differential antagonism by bicuculline and SR95531 of pentobarbitone-induced currents in cultured hippocampal neurons.

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The location of the gate in the acetylcholine receptor channel.

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Nicotinic receptors at the amino acid level

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Molecular dissection of benzodiazepine binding and allosteric coupling using chimeric gamma-aminobutyric acidA receptor subunits.

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Piperidine-4-sulphonic acid, a new specific GABA agonist

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Potassium currents expressed from Drosophila and mouse eag cDNAs in Xenopus oocytes.

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Pharmacology of barbiturate tolerance/dependence: GABAA receptors and molecular aspects

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State-dependent accessibility and electrostatic potential in the channel of the acetylcholine receptor. Inferences from rates of reaction of thiosulfonates with substituted cysteines in the M2 segment of the alpha subunit

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12 December 2020

Identification of benzodiazepine binding site residues in the gamma2 subunit of the gamma-aminobutyric acid(A) receptor

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12 December 2020

Single channel currents activated by gamma-aminobutyric acid, muscimol, and (-)-pentobarbital in cultured mouse spinal neurons

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Barbiturate interactions at the human GABAA receptor: dependence on receptor subunit combination

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Mapping the binding-site crevice of the dopamine D2 receptor by the substituted-cysteine accessibility method

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12 December 2020

Identification of amino acid residues of the NR2A subunit that control glutamate potency in recombinant NR1/NR2A NMDA receptors

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12 December 2020

Substituted-cysteine accessibility method

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12 December 2020

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

12 December 2020

Identification of channel-lining residues in the M2 membrane-spanning segment of the GABA(A) receptor alpha1 subunit

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12 December 2020

Nicotinic acetylcholine receptor at 4.6 A resolution: transverse tunnels in the channel wall.

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12 December 2020

Subunit stoichiometry of a mammalian K+ channel determined by construction of multimeric cDNAs.

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Interaction at End-Plate Receptors between Different Choline Derivatives

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12 December 2020

Identification of a [3H]muscimol photoaffinity substrate in the bovine gamma-aminobutyric acidA receptor alpha subunit.

1 reference

12 December 2020

Negatively charged amino acid residues in the nicotinic receptor delta subunit that contribute to the binding of acetylcholine

1 reference

12 December 2020

10.1523/JNEUROSCI.21-01-00067.2001

Identifiers

DOI

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3 November 2019

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3 November 2019

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