Distinct Molecular Recognition of Psychostimulants by Human andDrosophilaSerotonin Transporters (Q33194408)

23 July 2017

title

Distinct molecular recognition of psychostimulants by human and Drosophila serotonin transporters (English)

1 reference

23 July 2017

Distinct Molecular Recognition of Psychostimulants by Human andDrosophilaSerotonin Transporters (English)

1 reference

https://api.crossref.org/works/10.1124/JPET.103.057836

27 March 2024

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27 March 2024

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27 March 2024

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27 March 2024

author name string

David L. Roman

1

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27 March 2024

Shannon N. Saldaña

2

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27 March 2024

David E. Nichols

3

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27 March 2024

F. Ivy Carroll

4

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27 March 2024

Eric L. Barker

5

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27 March 2024

language of work or name

English

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publication date

30 October 2003

1 reference

full work available at URL

23 July 2017

https://syndication.highwire.org/content/doi/10.1124/jpet.103.057836

1 reference

https://api.crossref.org/works/10.1124/JPET.103.057836

Journal of Pharmacology and Experimental Therapeutics

27 March 2024

published in

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23 July 2017

volume

308

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23 July 2017

issue

2

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23 July 2017

page(s)

679-687

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Interactions of tryptamine derivatives with serotonin transporter species variants implicate transmembrane domain I in substrate recognition

23 July 2017

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Transmembrane domain I contributes to the permeation pathway for serotonin and ions in the serotonin transporter.

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High affinity recognition of serotonin transporter antagonists defined by species-scanning mutagenesis. An aromatic residue in transmembrane domain I dictates species-selective recognition of citalopram and mazindol

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Synthesis and transporter binding properties of 3beta-[4'-(phenylalkyl, -phenylalkenyl, and -phenylalkynyl)phenyl]tropane-2beta-carboxylic acid methyl esters: evidence of a remote phenyl binding domain on the dopamine transporter

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Synthesis, ligand binding, QSAR, and CoMFA study of 3 beta-(p-substituted phenyl)tropane-2 beta-carboxylic acid methyl esters

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A cocaine-sensitive Drosophila serotonin transporter: cloning, expression, and electrophysiological characterization

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Inhibition of plasma membrane monoamine transporters by beta-ketoamphetamines

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Cloning, expression, and localization of a chloride-facilitated, cocaine-sensitive serotonin transporter from Drosophila melanogaster

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Non-amines, drugs without an amine nitrogen, potently block serotonin transport: novel antidepressant candidates?

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Cloning of a serotonin transporter affected by antidepressants

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Psychostimulant-like effects of p-fluoroamphetamine in the rat

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N-substituted analogs of 2 beta-carbomethoxy-3 beta- (4'-iodophenyl)tropane (beta-CIT) with selective affinity to dopamine or serotonin transporters in rat forebrain.

27 March 2024

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Distinct recognition of substrates by the human and Drosophila serotonin transporters

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Identifiers

1 reference

23 July 2017

1 reference