A strategy to discover inhibitors of Bacillus subtilis surfactin-type phosphopantetheinyl transferase (Q33525922)

27 July 2017

title

A strategy to discover inhibitors of Bacillus subtilis surfactin-type phosphopantetheinyl transferase (English)

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27 July 2017

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Adam Yasgar

1

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Ajit Jadhav

object named as

Ajit Jadhav

3

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Anton Simeonov

6

object named as

Anton Simeonov

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27 July 2017

Timothy L Foley

2

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27 July 2017

James Inglese

4

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27 July 2017

Michael D Burkart

5

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27 July 2017

publication date

13 October 2009

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27 July 2017

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27 July 2017

volume

6

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27 July 2017

issue

2

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27 July 2017

page(s)

365-375

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A homogeneous resonance energy transfer assay for phosphopantetheinyl transferase

27 July 2017

cites work

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A robotic platform for quantitative high-throughput screening

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Compound Management for Quantitative High-Throughput Screening

21 June 2018

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High-throughput screening assays for the identification of chemical probes

21 June 2018

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Quantitative high-throughput screening: a titration-based approach that efficiently identifies biological activities in large chemical libraries

21 June 2018

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The nonredundant roles of two 4'-phosphopantetheinyl transferases in vital processes of Mycobacteria

21 June 2018

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Multiparameter analysis of a screen for progesterone receptor ligands: comparing fluorescence lifetime and fluorescence polarization measurements

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The 'allosteric modulator' SCH-202676 disrupts G protein-coupled receptor function via sulphydryl-sensitive mechanisms.

21 June 2018

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Genetically encoded short peptide tag for versatile protein labeling by Sfp phosphopantetheinyl transferase

21 June 2018

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21 June 2018

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21 June 2018

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Simultaneous determination of doxorubicin, daunorubicin, and idarubicin by capillary electrophoresis with laser-induced fluorescence detection

21 June 2018

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21 June 2018

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21 June 2018

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A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

21 June 2018

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Differential antiproliferative and apoptotic response of sanguinarine for cancer cells versus normal cells

21 June 2018

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Preparation of insoluble transmembrane peptides: glycophorin-A, prion (110-137), and FGFR (368-397).

21 June 2018

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21 June 2018

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21 June 2018

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A new enzyme superfamily - the phosphopantetheinyl transferases

21 June 2018

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Inhibition of HIV-1 infectivity by zinc-ejecting aromatic C-nitroso compounds

21 June 2018

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Cloning, overproduction, and characterization of the Escherichia coli holo-acyl carrier protein synthase

21 June 2018

1 reference

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Structure elucidation of Sch 538415, a novel acyl carrier protein synthase inhibitor from a microorganism

21 June 2018

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Anthranilate 4H-oxazol-5-ones: novel small molecule antibacterial acyl carrier protein synthase (AcpS) inhibitors.

21 January 2018

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Use of structure-based drug design approaches to obtain novel anthranilic acid acyl carrier protein synthase inhibitors

21 January 2018

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Manipulation of carrier proteins in antibiotic biosynthesis

21 January 2018

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DNA cleavage assay for the identification of topoisomerase I inhibitors

21 January 2018

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A high-throughput screen for aggregation-based inhibition in a large compound library

21 January 2018

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LPS inhibitors: key to overcoming multidrug-resistant bacteria?

21 January 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/20094656

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Biochemical and molecular analyses of the Streptococcus pneumoniae acyl carrier protein synthase, an enzyme essential for fatty acid biosynthesis

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20094656

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Characterization of Sfp, a Bacillus subtilis phosphopantetheinyl transferase for peptidyl carrier protein domains in peptide synthetases

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20094656

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1039/B913291K

1 reference

27 July 2017

1 reference

27 July 2017

1 reference