Divergent transducer-specific molecular efficacies generate biased agonism at a G protein-coupled receptor (GPCR) (Q33619504)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24668815%20AND%20SRC:MED&resulttype=core&format=json

12 March 2020

title

Divergent transducer-specific molecular efficacies generate biased agonism at a G protein-coupled receptor (GPCR) (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24668815%20AND%20SRC:MED&resulttype=core&format=json

G protein-coupled receptor

12 March 2020

main subject

0 references

author

Tommaso Costa

9

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12 March 2020

6

Alex Rojas Bie Thomsen

1 reference

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12 March 2020

10

Robert J Lefkowitz

1 reference

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12 March 2020

1

Ryan T Strachan

1 reference

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12 March 2020

author name string

Jin-peng Sun

2

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12 March 2020

David H Rominger

3

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12 March 2020

Jonathan D Violin

4

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12 March 2020

Seungkirl Ahn

5

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12 March 2020

Xiao Zhu

7

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12 March 2020

Andrew Kleist

8

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12 March 2020

language of work or name

English

0 references

publication date

25 March 2014

1 reference

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Journal of Biological Chemistry

12 March 2020

published in

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12 March 2020

volume

289

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issue

20

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12 March 2020

page(s)

14211-14224

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The β-arrestin-biased ligand TRV120023 inhibits angiotensin II-induced cardiac hypertrophy while preserving enhanced myofilament response to calcium

12 March 2020

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21 January 2018

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21 January 2018

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Side-chain substitutions within angiotensin II reveal different requirements for signaling, internalization, and phosphorylation of type 1A angiotensin receptors.

21 January 2018

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Promiscuous coupling at receptor-Galpha fusion proteins. The receptor of one covalent complex interacts with the alpha-subunit of another

21 January 2018

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Distinct phosphorylation sites on the β(2)-adrenergic receptor establish a barcode that encodes differential functions of β-arrestin.

21 January 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/24668815

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1074/JBC.M114.548131

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24668815%20AND%20SRC:MED&resulttype=core&format=json

12 March 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24668815%20AND%20SRC:MED&resulttype=core&format=json

12 March 2020

PubMed publication ID

24668815

1 reference

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