Fragment-based domain shuffling approach for the synthesis of pyran-based macrocycles (Q33839095)

29 July 2017

title

Fragment-based domain shuffling approach for the synthesis of pyran-based macrocycles (English)

1 reference

29 July 2017

Eamon Comer

1

1 reference

29 July 2017

Haibo Liu

2

1 reference

29 July 2017

Adrien Joliton

3

1 reference

29 July 2017

Alexandre Clabaut

4

1 reference

29 July 2017

Christopher Johnson

5

1 reference

29 July 2017

Lakshmi B Akella

6

1 reference

29 July 2017

Lisa A Marcaurelle

7

1 reference

29 July 2017

language of work or name

English

0 references

publication date

7 March 2011

1 reference

Proceedings of the National Academy of Sciences of the United States of America

29 July 2017

published in

1 reference

29 July 2017

volume

108

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29 July 2017

issue

17

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29 July 2017

page(s)

6751-6756

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Grand challenge commentary: Accessing new chemical space for 'undruggable' targets

29 July 2017

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28 July 2018

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Small molecules of different origins have distinct distributions of structural complexity that correlate with protein-binding profiles

28 July 2018

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Total synthesis of (-)-callipeltoside A

28 July 2018

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Factors determining the selection of organic reactions by medicinal chemists and the use of these reactions in arrays (small focused libraries).

28 July 2018

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Nitrile-containing pharmaceuticals: efficacious roles of the nitrile pharmacophore

28 July 2018

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28 July 2018

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Syntheses of aminoalcohol-derived macrocycles leading to a small-molecule binder to and inhibitor of Sonic Hedgehog

28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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Synthesis of a 35-member stereoisomer library of bistramide A: evaluation of effects on actin state, cell cycle and tumor cell growth

28 July 2018

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28 July 2018

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28 July 2018

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The interdependence between screening methods and screening libraries.

28 July 2018

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Synthesis of a library of complex macrodiolides employing cyclodimerization of hydroxy esters

28 July 2018

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Convergent synthesis of a complex oxime library using chemical domain shuffling

28 July 2018

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28 July 2018

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Fluorous mixture synthesis of stereoisomer libraries: total syntheses of (+)-murisolin and fifteen diastereoisomers

28 July 2018

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Molecular shape diversity of combinatorial libraries: a prerequisite for broad bioactivity.

28 July 2018

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Property distributions: differences between drugs, natural products, and molecules from combinatorial chemistry

28 July 2018

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The chemistry and biology of the bryostatin antitumour macrolides

28 July 2018

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28 July 2018

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28 July 2018

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Matrix assisted synthetic transformations: a mosaic of diverse contributions. II. The pattern is completed

28 July 2018

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Chemistry and Biology of the Immunophilins and Their Immunosuppressive Ligands

28 July 2018

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Escape from flatland: increasing saturation as an approach to improving clinical success.

28 July 2018

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Crossref

https://api.crossref.org/works/10.1073%2FPNAS.1015255108

Synthesis of all 16 stereoisomers of pinesaw fly sex pheromones--tools and tactics for solving problems in fluorous mixture synthesis.

21 January 2018

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Large-scale synthesis of all stereoisomers of a 2,3-unsaturated C-glycoside scaffold

21 January 2018

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Molecular diversity by design

29 October 2018

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Crossref

https://api.crossref.org/works/10.1073%2FPNAS.1015255108

Relationship of stereochemical and skeletal diversity of small molecules to cellular measurement space

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21383141

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Macrocycloadditions leading to conformationally restricted small molecules

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21383141

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Spongistatins, Cynachyrolides, or Altohyrtins? Marine Macrolides in Cancer Therapy

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21383141

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1073/PNAS.1015255108

1 reference

29 July 2017

0 references

1 reference

29 July 2017

1 reference