Aminoindoles, a novel scaffold with potent activity against Plasmodium falciparum (Q33851108)

29 July 2017

Aminoindoles, a novel scaffold with potent activity against Plasmodium falciparum (English)

1 reference

29 July 2017

Plasmodium falciparum

0 references

34

Dyann F Wirth

1 reference

29 July 2017

3

Ralph Mazitschek

0 references

Jingwen Lin

Jing-Wen Lin

14

0 references

Shahid M Khan

Shahid M Khan

16

0 references

Chris J Janse

Chris J Janse

15

0 references

Sergio Wittlin

25

Sergio Wittlin

1 reference

29 July 2017

17

Manoj Duraisingh

1 reference

29 July 2017

5

Renato Skerlj

1 reference

29 July 2017

10

Amar Bir Sidhu

1 reference

29 July 2017

4

Cassandra Celatka

1 reference

29 July 2017

Jose E Guerrero Bravo

11

Jose E Guerrero-Bravo

1 reference

29 July 2017

12

Keila N Crespo-Llado

1 reference

29 July 2017

13

Adelfa E Serrano

1 reference

29 July 2017

Maria Belen Jimenez-Diaz

20

María Belén Jiménez-Díaz

1 reference

29 July 2017

Petros Papastogiannidis

26

Petros Papastogiannidis

1 reference

29 July 2017

18

Bradley I Coleman

1 reference

29 July 2017

28

Jeffrey D Klinger

1 reference

29 July 2017

37

Edmund Sybertz

1 reference

29 July 2017

35

Jon Clardy

1 reference

29 July 2017

Robert H Barker

1

1 reference

29 July 2017

Sameer Urgaonkar

2

1 reference

29 July 2017

Ralph Mazitschek

3

1 reference

29 July 2017

Joseph F Cortese

6

1 reference

29 July 2017

Erin Tyndall

7

1 reference

29 July 2017

Hanlan Liu

8

1 reference

29 July 2017

Mandy Cromwell

9

1 reference

29 July 2017

Inigo Angulo-Barturen

19

1 reference

29 July 2017

Noemí Magán

21

1 reference

29 July 2017

Vanesa Gomez

22

1 reference

29 July 2017

Santiago Ferrer

23

1 reference

29 July 2017

María Santos Martínez

24

1 reference

29 July 2017

Thomas O'Shea

27

1 reference

29 July 2017

Mark Bree

29

1 reference

29 July 2017

Edward Lee

30

1 reference

29 July 2017

Mikaela Levine

31

1 reference

29 July 2017

Roger C Wiegand

32

1 reference

29 July 2017

Benito Munoz

33

1 reference

29 July 2017

Ian Bathurst

36

1 reference

29 July 2017

language of work or name

English

0 references

publication date

21 March 2011

1 reference

Antimicrobial Agents and Chemotherapy

29 July 2017

1 reference

29 July 2017

55

1 reference

29 July 2017

6

1 reference

29 July 2017

2612-2622

1 reference

Artemisinin‐induced dormancy in plasmodium falciparum: duration, recovery rates, and implications in treatment failure

29 July 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Spiroindolones, a potent compound class for the treatment of malaria

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Co-infections with Plasmodium knowlesi and other malaria parasites, Myanmar

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Novel Inhibitors of Plasmodium falciparum Dihydroorotate Dehydrogenase with Anti-malarial Activity in the Mouse Model

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Artemisinin Resistance in Plasmodium falciparum Malaria

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Improved murine model of malaria using Plasmodium falciparum competent strains and non-myelodepleted NOD-scid IL2Rgammanull mice engrafted with human erythrocytes

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Identification and characterization of small molecule inhibitors of a class I histone deacetylase from Plasmodium falciparum

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Comparative genomics of the neglected human malaria parasite Plasmodium vivax

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

In silico activity profiling reveals the mechanism of action of antimalarials discovered in a high-throughput screen

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

A murine model of falciparum-malaria by in vivo selection of competent strains in non-myelodepleted mice engrafted with human erythrocytes

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Malaria: progress, perils, and prospects for eradication

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

High-efficiency transfection and drug selection of genetically transformed blood stages of the rodent malaria parasite Plasmodium berghei

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Specific role of mitochondrial electron transport in blood-stage Plasmodium falciparum

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

High-throughput Plasmodium falciparum growth assay for malaria drug discovery

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

A Plasmodium berghei reference line that constitutively expresses GFP at a high level throughout the complete life cycle

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

DRUG RESISTANCE IN PLASMODIUM FALCIPARUM FROM THAILAND.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Chloroquine resistance in Plasmodium falciparum

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Malaria parasites giving rise to recrudescence in vitro

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Plasmodium knowlesi provides a rapid in vitro and in vivo transfection system that enables double-crossover gene knockout studies

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Pharmacokinetic interactions of antimalarial agents

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Identification of the human cytochrome P450 enzymes involved in the in vitro metabolism of artemisinin

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Resistance mutations reveal the atovaquone-binding domain of cytochrome b in malaria parasites

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Assessment of the effect of malaria infection on hepatic clearance of dihydroartemisinin using rat liver perfusions and microsomes

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Evidence of cross-contamination among laboratory lines of Plasmodium berghei

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Identification of human cytochrome P450 isoforms involved in the 3-hydroxylation of quinine by human live microsomes and nine recombinant human cytochromes P450

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

In vitro proguanil activation to cycloguanil by human liver microsomes is mediated by CYP3A isoforms as well as by S-mephenytoin hydroxylase

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Fansidar-resistant Plasmodium falciparum infection from Tanzania.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Effect of Plasmodium falciparum malaria infection on the plasma concentration of alpha 1-acid glycoprotein and the binding of quinine in Malawian children

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

The chemotherapy of rodent malaria, XXII. The value of drug-resistant strains of P. berghei in screening for blood schizontocidal activity

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

A concise silylamine approach to 2-amino-3-hydroxy-indoles with potent in vivo antimalaria activity

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Quantitative measurement of Plasmodium-infected erythrocytes in murine models of malaria by flow cytometry using bidimensional assessment of SYTO-16 fluorescence.

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Simple and sensitive antimalarial drug screening in vitro and in vivo using transgenic luciferase expressing Plasmodium berghei parasites.

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Improvement of detection specificity of Plasmodium-infected murine erythrocytes by flow cytometry using autofluorescence and YOYO-1.

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Plasmodium berghei: the application of cultivation and purification techniques to molecular studies of malaria parasites.

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Changes in susceptibility of Plasmodium falciparum to artesunate in vitro in Yunnan Province, China

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3101419

Frequency distribution of dapsone N-hydroxylase, a putative probe for P4503A4 activity, in a white population

29 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21422215

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Prediction of human pharmacokinetics from preclinical information: comparative accuracy of quantitative prediction approaches

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21422215

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1128/AAC.01714-10

1 reference

29 July 2017

1 reference

29 July 2017

1 reference