Pharmacological properties of a new antimalarial bisthiazolium salt, T3, and a corresponding prodrug, TE3. (Q33935408)

30 July 2017

title

Pharmacological properties of a new antimalarial bisthiazolium salt, T3, and a corresponding prodrug, TE3. (English)

1 reference

30 July 2017

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Olivier Nicolas

1

1 reference

30 July 2017

Delphine Margout

2

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30 July 2017

Nicolas Taudon

3

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30 July 2017

Sharon Wein

4

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30 July 2017

Michèle Calas

5

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30 July 2017

Henri J Vial

6

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30 July 2017

Françoise M M Bressolle

7

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30 July 2017

language of work or name

English

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publication date

1 September 2005

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Antimicrobial Agents and Chemotherapy

30 July 2017

published in

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30 July 2017

volume

49

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30 July 2017

issue

9

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30 July 2017

page(s)

3631-3639

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Prodrugs of bisthiazolium salts are orally potent antimalarials

30 July 2017

cites work

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5 July 2018

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Potent inhibitors of Plasmodium phospholipid metabolism with a broad spectrum of in vitro antimalarial activities

5 July 2018

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Heme binding contributes to antimalarial activity of bis-quaternary ammoniums

5 July 2018

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5 July 2018

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Medical need, scientific opportunity and the drive for antimalarial drugs

5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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Lipids and the malarial parasite

5 July 2018

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5 July 2018

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5 July 2018

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Liquid chromatography-electrospray mass spectrometry determination of a bis-thiazolium compound with potent antimalarial activity and its neutral bioprecursor in human plasma, whole blood and red blood cells

5 July 2018

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Quantification of antimalarial bisthiazolium compounds and their neutral bioprecursors in plasma by liquid chromatography-electrospray mass spectrometry

29 October 2018

1 reference

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29 October 2018

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Antimalarial activity of compounds interfering with Plasmodium falciparum phospholipid metabolism: comparison between mono- and bisquaternary ammonium salts

29 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/16127032

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Modelling of individual pharmacokinetics for computer-aided drug dosage

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/16127032

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1128/AAC.49.9.3631-3639.2005

1 reference

release_rvvwft6nxzat3m2qxblhxpg4e4

30 July 2017

Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/rvvwft6nxzat3m2qxblhxpg4e4

mapped directly with Wikidata item

24 November 2022

based on heuristic

PMC publication ID

1195427

1 reference

30 July 2017

1 reference