Assessing subunit dependency of the Plasmodium proteasome using small molecule inhibitors and active site probes (Q34061291)

30 July 2017

Assessing subunit dependency of the Plasmodium proteasome using small molecule inhibitors and active site probes (English)

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30 July 2017

Martijn Verdoes

3

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Herman S Overkleeft

object named as

Herman S Overkleeft

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Matthew Bogyo

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object named as

Matthew Bogyo

1 reference

30 July 2017

5

Fiona E McAllister

1 reference

30 July 2017

Hao Li

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30 July 2017

Wouter A van der Linden

2

1 reference

30 July 2017

Bogdan I Florea

4

1 reference

30 July 2017

Kavitha Govindaswamy

6

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30 July 2017

Joshua E Elias

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30 July 2017

Purnima Bhanot

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30 July 2017

language of work or name

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19 June 2014

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30 July 2017

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30 July 2017

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30 July 2017

1869-1876

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describes a project that uses

30 July 2017

ImageJ

1 reference

11 June 2022

https://www.ebi.ac.uk/europepmc/webservices/rest/PMC4136710/fullTextXML

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28 July 2018

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28 July 2018

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Quiescent fibroblasts are protected from proteasome inhibition-mediated toxicity

28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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Specific cell-permeable inhibitor of proteasome trypsin-like sites selectively sensitizes myeloma cells to bortezomib and carfilzomib

28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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Selective inhibitor of proteasome's caspase-like sites sensitizes cells to specific inhibition of chymotrypsin-like sites

28 July 2018

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28 July 2018

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28 July 2018

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Extensive immunoglobulin production sensitizes myeloma cells for proteasome inhibition.

28 July 2018

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A fluorescent broad-spectrum proteasome inhibitor for labeling proteasomes in vitro and in vivo

28 July 2018

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How many functional transport pathways does Plasmodium falciparum induce in the membrane of its host erythrocyte?

28 July 2018

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The transcriptome of the intraerythrocytic developmental cycle of Plasmodium falciparum

28 July 2018

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Inhibition of proteasome activity induces concerted expression of proteasome genes and de novo formation of Mammalian proteasomes

28 July 2018

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28 July 2018

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The catalytic sites of 20S proteasomes and their role in subunit maturation: a mutational and crystallographic study

28 July 2018

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Proteasome inhibitors block development of Plasmodium spp.

28 July 2018

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The active sites of the eukaryotic 20 S proteasome and their involvement in subunit precursor processing

28 July 2018

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Identification of the yeast 20S proteasome catalytic centers and subunit interactions required for active-site formation

28 July 2018

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Autocatalytic subunit processing couples active site formation in the 20S proteasome to completion of assembly

28 July 2018

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Incorporation of Non-natural Amino Acids Improves Cell Permeability and Potency of Specific Inhibitors of Proteasome Trypsin-like Sites

28 July 2018

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Nature of pharmacophore influences active site specificity of proteasome inhibitors

28 October 2018

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Marine actinomycetes: a new source of compounds against the human malaria parasite

28 October 2018

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28 October 2018

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Importance of the different proteolytic sites of the proteasome and the efficacy of inhibitors varies with the protein substrate

28 October 2018

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PubMed

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12 December 2020

based on heuristic

Identifiers

DOI

10.1021/CB5001263

1 reference

30 July 2017

1 reference

30 July 2017

1 reference