Pharmacophore-based virtual screening and biological evaluation of small molecule inhibitors for protein arginine methylation (Q34113450)

31 July 2017

title

Pharmacophore-based virtual screening and biological evaluation of small molecule inhibitors for protein arginine methylation (English)

1 reference

31 July 2017

1 reference

Juxian Wang

1

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31 July 2017

Limin Chen

2

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31 July 2017

Sarmistha Halder Sinha

3

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31 July 2017

Zhongjie Liang

4

1 reference

31 July 2017

Huifang Chai

5

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31 July 2017

Sakthivel Muniyan

6

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31 July 2017

Yu-Wei Chou

7

1 reference

31 July 2017

Chao Yang

8

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31 July 2017

Leilei Yan

9

1 reference

31 July 2017

You Feng

10

1 reference

31 July 2017

Keqin Kathy Li

11

1 reference

31 July 2017

Ming-Fong Lin

12

1 reference

31 July 2017

Hualiang Jiang

13

1 reference

31 July 2017

Yujun George Zheng

14

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31 July 2017

Cheng Luo

15

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31 July 2017

language of work or name

English

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publication date

12 September 2012

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Journal of Medicinal Chemistry

31 July 2017

published in

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31 July 2017

volume

55

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31 July 2017

issue

18

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31 July 2017

page(s)

7978-7987

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Chemical and biochemical approaches in the study of histone methylation and demethylation

31 July 2017

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1 reference

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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Virtual screening and biological characterization of novel histone arginine methyltransferase PRMT1 inhibitors

5 July 2018

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5 July 2018

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epigenetic multiple ligands: mixed histone/protein methyltransferase, acetyltransferase, and class III deacetylase (sirtuin) inhibitors.

5 July 2018

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A glycine-arginine domain in control of the human MRE11 DNA repair protein

5 July 2018

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5 July 2018

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Protein arginine-methyltransferase-dependent oncogenesis

5 July 2018

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A novel arginine methyltransferase inhibitor with cellular activity

5 July 2018

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Target-based approach to inhibitors of histone arginine methyltransferases

5 July 2018

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Small molecule inhibitors of histone arginine methyltransferases: homology modeling, molecular docking, binding mode analysis, and biological evaluations

5 July 2018

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Histone arginine methylation regulates pluripotency in the early mouse embryo

5 July 2018

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5 July 2018

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Chromatin modifications as targets for new anticancer drugs

5 July 2018

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Arginine methylation an emerging regulator of protein function

5 July 2018

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Pharmacophore modeling and three dimensional database searching for drug design using catalyst: recent advances

5 July 2018

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Small molecule regulators of protein arginine methyltransferases

5 July 2018

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The antifungal antibiotic sinefungin as a ver y active inhibitor of methyltransferases and of the transformation of chick embryo fibroblasts by rous sarcoma virus

5 July 2018

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3D-QSAR based pharmacophore modeling and virtual screening for identification of novel pteridine reductase inhibitors.

5 July 2018

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Discovery and mechanistic study of a class of protein arginine methylation inhibitors.

28 October 2018

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A dual-mode fluorescence strategy for screening HAT modulators

28 October 2018

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Bisubstrate Inhibitors of the MYST HATs Esa1 and Tip60.

28 October 2018

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Role of asymmetric dimethylarginine in inflammatory reactions by angiotensin II.

28 October 2018

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Establishment and characterization of androgen-independent human prostate cancer LNCaP cell model

28 October 2018

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Transcriptional coactivator protein p300. Kinetic characterization of its histone acetyltransferase activity

28 October 2018

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Expression of human prostatic acid phosphatase correlates with androgen-stimulated cell proliferation in prostate cancer cell lines

28 October 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/22928876

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Multiple pharmacophore models combined with molecular docking: a reliable way for efficiently identifying novel PDE4 inhibitors with high structural diversity

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22928876

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/JM300521M

1 reference

31 July 2017

1 reference

31 July 2017

1 reference