Synthesis, biological evaluation, and structure-activity relationships of a novel class of apurinic/apyrimidinic endonuclease 1 inhibitors (Q34210627)

31 July 2017

Synthesis, biological evaluation, and structure-activity relationships of a novel class of apurinic/apyrimidinic endonuclease 1 inhibitors (English)

1 reference

31 July 2017

Ajit Jadhav

5

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Anton Simeonov

4

object named as

Anton Simeonov

1 reference

31 July 2017

Ganesha Rai

1

1 reference

31 July 2017

Vaddadi N Vyjayanti

2

1 reference

31 July 2017

Dorjbal Dorjsuren

3

1 reference

31 July 2017

David M Wilson

6

1 reference

31 July 2017

David J Maloney

7

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31 July 2017

language of work or name

English

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publication date

28 March 2012

1 reference

Journal of Medicinal Chemistry

31 July 2017

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31 July 2017

55

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31 July 2017

7

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31 July 2017

3101-3112

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describes a project that uses

31 July 2017

ImageQuant

1 reference

11 June 2022

https://www.ebi.ac.uk/europepmc/webservices/rest/PMC3515842/fullTextXML

based on heuristic

inferred from PubMed Central ID database lookup

cites work

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Novel small-molecule inhibitor of apurinic/apyrimidinic endonuclease 1 blocks proliferation and reduces viability of glioblastoma cells

5 July 2018

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PARP inhibition: PARP1 and beyond

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5 July 2018

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Identification and characterization of inhibitors of human apurinic/apyrimidinic endonuclease APE1

5 July 2018

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The many functions of APE1/Ref-1: not only a DNA repair enzyme

5 July 2018

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Transcriptional regulatory functions of mammalian AP-endonuclease (APE1/Ref-1), an essential multifunctional protein

5 July 2018

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Potent inhibition of human apurinic/apyrimidinic endonuclease 1 by arylstibonic acids

5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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Molecular and biological roles of Ape1 protein in mammalian base excision repair

5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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Inhibition of the human apurinic/apyrimidinic endonuclease (APE1) repair activity and sensitization of breast cancer cells to DNA alkylating agents with lucanthone.

5 July 2018

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Discovery and SAR of a novel selective and orally bioavailable nonpeptide classical competitive inhibitor class of protein-tyrosine phosphatase 1B.

5 July 2018

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The major human abasic endonuclease: formation, consequences and repair of abasic lesions in DNA.

5 July 2018

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Elements in abasic site recognition by the major human and Escherichia coli apurinic/apyrimidinic endonucleases

5 July 2018

1 reference

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Topoisomerase inhibition by lucanthone, an adjuvant in radiation therapy

5 July 2018

1 reference

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Abasic site binding by the human apurinic endonuclease, Ape, and determination of the DNA contact sites

5 July 2018

1 reference

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Repair of oxidative damage to DNA: enzymology and biology

5 July 2018

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Incision activity of human apurinic endonuclease (Ape) at abasic site analogs in DNA

5 July 2018

1 reference

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Pharmacophore guided discovery of small-molecule human apurinic/apyrimidinic endonuclease 1 inhibitors

5 July 2018

1 reference

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Apurinic/apyrimidinic endonuclease activity is elevated in human adult gliomas.

28 October 2018

1 reference

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Methoxyamine potentiates DNA single strand breaks and double strand breaks induced by temozolomide in colon cancer cells

28 October 2018

1 reference

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28 October 2018

Identifiers

DOI

10.1021/JM201537D

1 reference

31 July 2017

1 reference

31 July 2017

1 reference