Antinociceptive effects of the N-acylethanolamine acid amidase inhibitor ARN077 in rodent pain models (Q34315969)

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19 February 2020

title

Antinociceptive effects of the N-acylethanolamine acid amidase inhibitor ARN077 in rodent pain models (English)

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19 February 2020

10

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19 February 2020

Rosalia Bertorelli

11

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19 February 2020

author name string

Oscar Sasso

1

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19 February 2020

Guillermo Moreno-Sanz

2

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19 February 2020

Cataldo Martucci

3

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19 February 2020

Natalia Realini

4

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19 February 2020

Mauro Dionisi

5

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19 February 2020

Luisa Mengatto

6

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19 February 2020

Andrea Duranti

7

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19 February 2020

Glauco Tarozzo

8

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19 February 2020

Giorgio Tarzia

9

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19 February 2020

Angelo Reggiani

12

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19 February 2020

Daniele Piomelli

13

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19 February 2020

language of work or name

English

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publication date

2 November 2012

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19 February 2020

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19 February 2020

volume

154

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19 February 2020

issue

3

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19 February 2020

page(s)

350-360

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β-Lactones Inhibit N-acylethanolamine Acid Amidase by S-Acylation of the Catalytic N-Terminal Cysteine

19 February 2020

cites work

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Proinflammatory stimuli control N-acylphosphatidylethanolamine-specific phospholipase D expression in macrophages

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Synthesis and structure-activity relationships of N-(2-oxo-3-oxetanyl)amides as N-acylethanolamine-hydrolyzing acid amidase inhibitors.

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Selective N-acylethanolamine-hydrolyzing acid amidase inhibition reveals a key role for endogenous palmitoylethanolamide in inflammation.

6 July 2018

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Inhibition of fatty acid amide hydrolase produces PPAR-alpha-mediated analgesia in a rat model of inflammatory pain

6 July 2018

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Synergistic antinociception by the cannabinoid receptor agonist anandamide and the PPAR-alpha receptor agonist GW7647.

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Molecular characterization of N-acylethanolamine-hydrolyzing acid amidase, a novel member of the choloylglycine hydrolase family with structural and functional similarity to acid ceramidase

6 July 2018

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The nuclear receptor peroxisome proliferator-activated receptor-alpha mediates the anti-inflammatory actions of palmitoylethanolamide.

6 July 2018

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Oleylethanolamide regulates feeding and body weight through activation of the nuclear receptor PPAR-alpha

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Design, synthesis, and structure-activity relationships of alkylcarbamic acid aryl esters, a new class of fatty acid amide hydrolase inhibitors.

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Structural basis for antagonist-mediated recruitment of nuclear co-repressors by PPARalpha

6 July 2018

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28 October 2018

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28 October 2018

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28 October 2018

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1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/23218523

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

N-(2-Oxo-3-oxetanyl)carbamic Acid Esters as N-Acylethanolamine Acid Amidase Inhibitors: Synthesis and Structure–Activity and Structure–Property Relationships

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/23218523

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.PAIN.2012.10.018

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23218523%20AND%20SRC:MED&resulttype=core&format=json

19 February 2020

1 reference

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19 February 2020

PubMed publication ID

23218523

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23218523%20AND%20SRC:MED&resulttype=core&format=json