Trypanocidal furamidine analogues: influence of pyridine nitrogens on trypanocidal activity, transport kinetics, and resistance patterns (Q34933034)

5 August 2017

title

Trypanocidal furamidine analogues: influence of pyridine nitrogens on trypanocidal activity, transport kinetics, and resistance patterns (English)

1 reference

5 August 2017

5

Michael P Barrett

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Richard Burchmore

object named as

Richard J Burchmore

3

0 references

Harry P de Koning

object named as

Harry P de Koning

4

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author name string

Christopher P Ward

1

1 reference

5 August 2017

Pui Ee Wong

2

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5 August 2017

Michael P Barrett

5

1 reference

5 August 2017

language of work or name

English

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publication date

14 March 2011

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Antimicrobial Agents and Chemotherapy

5 August 2017

published in

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5 August 2017

volume

55

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5 August 2017

issue

5

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5 August 2017

page(s)

2352-2361

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A molecular mechanism for eflornithine resistance in African trypanosomes

5 August 2017

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8 July 2018

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8 July 2018

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8 July 2018

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8 July 2018

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8 July 2018

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8 July 2018

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8 July 2018

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26 October 2018

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26 October 2018

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26 October 2018

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Different substrate recognition motifs of human and trypanosome nucleobase transporters. Selective uptake of purine antimetabolites

26 October 2018

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Further evidence for a link between melarsoprol resistance and P2 transporter function in African trypanosomes.

26 October 2018

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A diamidine-resistant Trypanosoma equiperdum clone contains a P2 purine transporter with reduced substrate affinity.

26 October 2018

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Human African trypanosomiasis

26 October 2018

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Ever-increasing complexities of diamidine and arsenical crossresistance in African trypanosomes

9 December 2018

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Molecular Interactions Underlying the Unusually High Adenosine Affinity of a Novel Trypanosoma brucei Nucleoside Transporter

9 December 2018

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9 December 2018

12 December 2020

Time-dose-response of Trypanosoma brucei brucei to diminazene aceturate (Berenil) and in vitro simulation of drug-concentration-time profiles in cattle plasma

1 reference

12 December 2020

Purine stress in crithidia: adaptation of a parasite to environmental stress

1 reference

12 December 2020

Purine nucleobase transport in bloodstream forms of Trypanosoma brucei brucei is mediated by two novel transporters

1 reference

12 December 2020

Hypoxanthine uptake through a purine-selective nucleobase transporter in Trypanosoma brucei brucei procyclic cells is driven by protonmotive force

1 reference

12 December 2020

Differential regulation of nucleoside and nucleobase transporters in Crithidia fasciculata and Trypanosoma brucei brucei

1 reference

12 December 2020

Characterization of a Nucleoside/Proton Symporter in ProcyclicTrypanosoma brucei brucei

1 reference

12 December 2020

Adenosine transporters in bloodstream forms of Trypanosoma brucei brucei: substrate recognition motifs and affinity for trypanocidal drugs

1 reference

12 December 2020

Identifiers

DOI

10.1128/AAC.01551-10

1 reference

5 August 2017

1 reference

5 August 2017

1 reference