CP47,497-C8 and JWH073, commonly found in 'Spice' herbal blends, are potent and efficacious CB(1) cannabinoid receptor agonists (Q34981205)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21333643%20AND%20SRC:MED&resulttype=core&format=json

22 January 2020

title

CP47,497-C8 and JWH073, commonly found in 'Spice' herbal blends, are potent and efficacious CB(1) cannabinoid receptor agonists (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21333643%20AND%20SRC:MED&resulttype=core&format=json

22 January 2020

0 references

0 references

0 references

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21333643%20AND%20SRC:MED&resulttype=core&format=json

22 January 2020

Ken Mackie

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21333643%20AND%20SRC:MED&resulttype=core&format=json

22 January 2020

author name string

Donghoon Lee

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21333643%20AND%20SRC:MED&resulttype=core&format=json

22 January 2020

Alex Straiker

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21333643%20AND%20SRC:MED&resulttype=core&format=json

22 January 2020

Theodore S Widlanski

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21333643%20AND%20SRC:MED&resulttype=core&format=json

22 January 2020

language of work or name

English

0 references

publication date

16 February 2011

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21333643%20AND%20SRC:MED&resulttype=core&format=json

European Journal of Pharmacology

22 January 2020

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21333643%20AND%20SRC:MED&resulttype=core&format=json

22 January 2020

volume

659

1 reference

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22 January 2020

issue

2-3

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22 January 2020

page(s)

139-145

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21333643%20AND%20SRC:MED&resulttype=core&format=json

Spice drugs as a new trend: mode of action, identification and legislation

22 January 2020

cites work

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JWH018, a common constituent of 'Spice' herbal blends, is a potent and efficacious cannabinoid CB receptor agonist

8 July 2018

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Spice: a never ending story?

8 July 2018

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Rapid CB1 cannabinoid receptor desensitization defines the time course of ERK1/2 MAP kinase signaling.

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8 July 2018

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8 July 2018

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8 July 2018

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8 July 2018

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Cloning and molecular characterization of the rat CB2 cannabinoid receptor

8 July 2018

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8 July 2018

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Influence of the N-1 alkyl chain length of cannabimimetic indoles upon CB(1) and CB(2) receptor binding

8 July 2018

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Effects of the endogeneous cannabinoid, anandamide, on neuronal activity in rat hippocampal slices

8 July 2018

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Structure-activity relationships of indole- and pyrrole-derived cannabinoids

8 July 2018

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Evaluation of cannabinoid receptor agonists and antagonists using the guanosine-5'-O-(3-[35S]thio)-triphosphate binding assay in rat cerebellar membranes.

8 July 2018

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A cannabinoid derived prototypical analgesic

8 July 2018

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Excitatory and inhibitory autaptic currents in isolated hippocampal neurons maintained in cell culture

8 July 2018

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Pharmacological profile of a series of bicyclic cannabinoid analogs: classification as cannabimimetic agents

8 July 2018

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8 July 2018

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How globalization and market innovation challenge how we think about and respond to drug use: 'Spice' a case study.

8 July 2018

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26 October 2018

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26 October 2018

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26 October 2018

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26 October 2018

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26 October 2018

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A mutation in the second transmembrane region of the CB1 receptor selectively disrupts G protein signaling and prevents receptor internalization.

26 October 2018

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Distinct domains of the CB1 cannabinoid receptor mediate desensitization and internalization.

26 October 2018

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Cannabinoid receptor agonists inhibit glutamatergic synaptic transmission in rat hippocampal cultures.

26 October 2018

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Structure-activity relationships for cannabinoid receptor-binding and analgesic activity: studies of bicyclic cannabinoid analogs

26 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21333643

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Use of high-resolution accurate mass spectrometry to detect reported and previously unreported cannabinomimetics in "herbal high" products

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21333643

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Internalization and Recycling of the CB1 Cannabinoid Receptor

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21333643

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.EJPHAR.2011.01.066

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21333643%20AND%20SRC:MED&resulttype=core&format=json

22 January 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21333643%20AND%20SRC:MED&resulttype=core&format=json

22 January 2020

1 reference