Nobilamides A-H, long-acting transient receptor potential vanilloid-1 (TRPV1) antagonists from mollusk-associated bacteria (Q35097693)

6 August 2017

title

Nobilamides A-H, long-acting transient receptor potential vanilloid-1 (TRPV1) antagonists from mollusk-associated bacteria (English)

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Ac-Phe-D-Leu-Phe-D-aThr-Val-Ala-Abu(2,3-dehydro)-OH

6 August 2017

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8

Baldomero M Olivera

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6 August 2017

4

Ronald W Hughen

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6 August 2017

5

Lenny Marett

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6 August 2017

Zhenjian Lin

1

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6 August 2017

Christopher A Reilly

2

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6 August 2017

Rowena Antemano

3

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6 August 2017

Gisela P Concepcion

6

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6 August 2017

Margo G Haygood

7

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6 August 2017

Alan Light

9

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6 August 2017

Eric W Schmidt

10

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6 August 2017

language of work or name

English

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publication date

16 May 2011

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full work available at URL

6 August 2017

https://europepmc.org/articles/pmc3133741?pdf=render

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19 March 2024

https://api.unpaywall.org/v2/10.1021/jm101621u?email=unpaywall_01@example.com

published in

Journal of Medicinal Chemistry

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6 August 2017

volume

54

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6 August 2017

issue

11

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6 August 2017

page(s)

3746-3755

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https://api.unpaywall.org/v2/10.1021/jm101621u?email=unpaywall_01@example.com

6 August 2017

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19 March 2024

access restriction status

open access

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inferred from online access status

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Structure-activity relationship of capsaicin analogs and transient receptor potential vanilloid 1-mediated human lung epithelial cell toxicity

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The biophysical and molecular basis of TRPV1 proton gating

9 July 2018

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Pulicatins A-E, neuroactive thiazoline metabolites from cone snail-associated bacteria

9 July 2018

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International Union of Basic and Clinical Pharmacology. LXXVI. Current progress in the mammalian TRP ion channel family

9 July 2018

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A bivalent tarantula toxin activates the capsaicin receptor, TRPV1, by targeting the outer pore domain

9 July 2018

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TRPV1: on the road to pain relief

9 July 2018

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Oxidative challenges sensitize the capsaicin receptor by covalent cysteine modification

9 July 2018

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TRPV1 and TRPA1 mediate peripheral nitric oxide-induced nociception in mice

9 July 2018

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The endoplasmic reticulum of dorsal root ganglion neurons contains functional TRPV1 channels

9 July 2018

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Microhabitats within venomous cone snails contain diverse actinobacteria

9 July 2018

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Pore region of TRPV3 ion channel is specifically required for heat activation

9 July 2018

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Clinical development of TRPV1 antagonists: targeting a pivotal point in the pain pathway

9 July 2018

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Molecular modeling of the full-length human TRPV1 channel in closed and desensitized states.

9 July 2018

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A single N-terminal cysteine in TRPV1 determines activation by pungent compounds from onion and garlic

9 July 2018

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On the mechanism of TBA block of the TRPV1 channel.

9 July 2018

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Transient receptor potential vanilloid 1 agonists cause endoplasmic reticulum stress and cell death in human lung cells

9 July 2018

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TRP channel activation by reversible covalent modification

9 July 2018

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Reducing and oxidizing agents sensitize heat-activated vanilloid receptor (TRPV1) current

9 July 2018

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Calcium-dependent and independent mechanisms of capsaicin receptor (TRPV1)-mediated cytokine production and cell death in human bronchial epithelial cells

9 July 2018

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TRPV1 antagonists elevate cell surface populations of receptor protein and exacerbate TRPV1-mediated toxicities in human lung epithelial cells

9 July 2018

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Vanilloid receptor TRPV1 antagonists as the next generation of painkillers. Are we putting the cart before the horse?

9 July 2018

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Capsaicinoids Cause Inflammation and Epithelial Cell Death through Activation of Vanilloid Receptors

9 July 2018

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Chemistry, nutrition, and microbiology of D-amino acids.

9 July 2018

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The capsaicin receptor: a heat-activated ion channel in the pain pathway

9 July 2018

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Ser-His catalyses the formation of peptides and PNAs

9 July 2018

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Total synthesis of bacilosarcins A and B

27 September 2018

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12 December 2020

Isolation of a new peptide antibiotic TL-119. Studies on antibiotics from the genus Bacillus. IV

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12 December 2020

Revised structure of the peptide lactone antibiotic, TL-119 and/or A-3302-B

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12 December 2020

Nonribosomal Peptide Biosynthesis: Point Mutations and Module Skipping Lead to Chemical Diversity

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12 December 2020

Substance P released by TRPV1-expressing neurons produces reactive oxygen species that mediate ethanol-induced gastric injury

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12 December 2020

Identifiers

DOI

10.1021/JM101621U

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6 August 2017

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6 August 2017

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