Highly selective salicylketoxime-based estrogen receptor β agonists display antiproliferative activities in a glioma model (Q36175547)

12 August 2017

Highly selective salicylketoxime-based estrogen receptor β agonists display antiproliferative activities in a glioma model (English)

1 reference

12 August 2017

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25559213%20AND%20SRC:MED&resulttype=core&format=json

13 June 2020

Carlotta Granchi

3

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13 June 2020

Tiziano Tuccinardi

4

1 reference

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13 June 2020

Adriano Martinelli

6

1 reference

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13 June 2020

Isabella Caligiuri

7

1 reference

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13 June 2020

Giuseppe Toffoli

8

1 reference

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13 June 2020

Flavio Rizzolio

9

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13 June 2020

Filippo Minutolo

13

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13 June 2020

Benita Katzenellenbogen

11

object named as

Benita S Katzenellenbogen

1 reference

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13 June 2020

10

Kathryn E Carlson

1 reference

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13 June 2020

John A Katzenellenbogen

12

object named as

John A Katzenellenbogen

1 reference

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13 June 2020

1

Ilaria Paterni

1 reference

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13 June 2020

author name string

Marco Macchia

5

1 reference

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13 June 2020

language of work or name

English

0 references

publication date

14 January 2015

1 reference

Journal of Medicinal Chemistry

12 August 2017

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25559213%20AND%20SRC:MED&resulttype=core&format=json

13 June 2020

volume

58

1 reference

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13 June 2020

issue

3

1 reference

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13 June 2020

page(s)

1184-1194

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25559213%20AND%20SRC:MED&resulttype=core&format=json

Estrogen receptors alpha (ERα) and beta (ERβ): subtype-selective ligands and clinical potential.

13 June 2020

cites work

1 reference

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Mechanisms enforcing the estrogen receptor β selectivity of botanical estrogens

1 October 2017

1 reference

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Ligand-binding dynamics rewire cellular signaling via estrogen receptor-α

1 October 2017

1 reference

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Estrogen inhibits renal cell carcinoma cell progression through estrogen receptor-β activation

1 October 2017

1 reference

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Therapeutic significance of estrogen receptor β agonists in gliomas

1 October 2017

1 reference

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Selective and potent agonists for estrogen receptor beta derived from molecular refinements of salicylaldoximes.

1 October 2017

1 reference

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Estrogen receptor β exerts tumor repressive functions in human malignant pleural mesothelioma via EGFR inactivation and affects response to gefitinib

1 October 2017

1 reference

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Estrogen receptors: therapies targeted to receptor subtypes

1 October 2017

1 reference

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Do steroid hormones play a role in the etiology of glioma?

1 October 2017

1 reference

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Estrogen receptor-beta activated apoptosis in benign hyperplasia and cancer of the prostate is androgen independent and TNFalpha mediated

1 October 2017

1 reference

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Estrogen receptor β ligands: recent advances and biomedical applications.

1 October 2017

1 reference

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Genome-wide dynamics of chromatin binding of estrogen receptors alpha and beta: mutual restriction and competitive site selection

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4610302

AutoDock4 and AutoDockTools4: Automated docking with selective receptor flexibility

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4610302

Structural evolutions of salicylaldoximes as selective agonists for estrogen receptor beta

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4610302

Monoaryl-substituted salicylaldoximes as ligands for estrogen receptor beta

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4610302

Estrogen Receptors alpha and beta as determinants of gene expression: influence of ligand, dose, and chromatin binding

1 October 2017

1 reference

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International Union of Pharmacology. LXIV. Estrogen receptors

1 October 2017

1 reference

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Benzopyrans are selective estrogen receptor beta agonists with novel activity in models of benign prostatic hyperplasia

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4610302

Estrogen receptor (ER)-beta isoforms: a key to understanding ER-beta signaling

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4610302

Impact of estrogen receptor beta on gene networks regulated by estrogen receptor alpha in breast cancer cells

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4610302

Reproductive and hormonal factors and risk of brain tumors in adult females

1 October 2017

1 reference

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Reproductive factors and risk of glioma in women

1 October 2017

1 reference

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Reduced expression of oestrogen receptor β in invasive breast cancer and its re‐expression using DNA methyl transferase inhibitors in a cell line model

1 October 2017

1 reference

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1 October 2017

The Protein Data Bank

1 reference

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Estrogen receptor subtype-selective ligands: asymmetric synthesis and biological evaluation of cis- and trans-5,11-dialkyl- 5,6,11, 12-tetrahydrochrysenes

1 October 2017

1 reference

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Novel ligands that function as selective estrogens or antiestrogens for estrogen receptor-alpha or estrogen receptor-beta

1 October 2017

1 reference

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Tumor repressive functions of estrogen receptor beta in SW480 colon cancer cells.

1 October 2017

1 reference

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Altered ligand binding properties and enhanced stability of a constitutively active estrogen receptor: evidence that an open pocket conformation is required for ligand interaction.

2 July 2018

1 reference

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Photoaffinity labels for estrogen binding proteins of rat uterus.

2 July 2018

1 reference

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Synthesis of highly substituted pyrroles via nucleophilic catalysis

2 July 2018

1 reference

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C-H hydroxylation using a heterocyclic catalyst and aqueous H2O2.

23 September 2018

1 reference

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An efficient synthesis of a dual PPAR alpha/gamma agonist and the formation of a sterically congested alpha-aryloxyisobutyric acid via a Bargellini reaction

23 September 2018

1 reference

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Steroid hormone receptors in astrocytic neoplasms.

23 September 2018

1 reference

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O-Nucleophilic Amino Alcohol Acyl-Transfer Catalysts: the Effect of Acidity of the Hydroxyl Group on the Activity of the Catalyst

23 September 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/25559213

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/JM501829F

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25559213%20AND%20SRC:MED&resulttype=core&format=json

13 June 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25559213%20AND%20SRC:MED&resulttype=core&format=json

13 June 2020

1 reference