AM630 behaves as a protean ligand at the human cannabinoid CB2 receptor. (Q36176518)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21615724%20AND%20SRC:MED&resulttype=core&format=json

2 February 2020

title

AM630 behaves as a protean ligand at the human cannabinoid CB2 receptor (English)

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2 February 2020

0 references

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4

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2 February 2020

1

Daniele Bolognini

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2 February 2020

3

Daniela Parolaro

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2 February 2020

author name string

Maria Grazia Cascio

series ordinal

2

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2 February 2020

language of work or name

English

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publication date

1 April 2012

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British Journal of Pharmacology

2 February 2020

published in

1 reference

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2 February 2020

volume

165

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2 February 2020

issue

8

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2 February 2020

page(s)

2561-2574

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Guide to Receptors and Channels (GRAC), 5th edition

2 February 2020

cites work

1 reference

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International Union of Basic and Clinical Pharmacology. LXXIX. Cannabinoid receptors and their ligands: beyond CB₁ and CB₂

1 October 2017

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Evaluation of Cannabinoid Receptor 2 and Metabotropic Glutamate Receptor 1 Functional Responses Using a Cell Impedance–Based Technology

1 October 2017

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The plant cannabinoid Delta9-tetrahydrocannabivarin can decrease signs of inflammation and inflammatory pain in mice

1 October 2017

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Updating the chemistry and biology of cannabinoid CB2 receptor-specific inverse agonists

1 October 2017

1 reference

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Regulation of CB1 cannabinoid receptor trafficking by the adaptor protein AP-3

1 October 2017

1 reference

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Biology and therapeutic potential of cannabinoid CB2 receptor inverse agonists

1 October 2017

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G-protein-coupled receptors signalling at the cell nucleus: an emerging paradigm.

1 October 2017

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In vitro pharmacological characterization of AM1241: a protean agonist at the cannabinoid CB2 receptor?

1 October 2017

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Pharmacological actions of cannabinoids.

1 October 2017

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Evidence that the plant cannabinoid Delta9-tetrahydrocannabivarin is a cannabinoid CB1 and CB2 receptor antagonist

1 October 2017

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International Union of Pharmacology. XXVII. Classification of cannabinoid receptors

1 October 2017

1 reference

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Inverse, protean, and ligand-selective agonism: matters of receptor conformation

1 October 2017

1 reference

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Structural determinants of the partial agonist-inverse agonist properties of 6'-azidohex-2'-yne-delta8-tetrahydrocannabinol at cannabinoid receptors

1 October 2017

1 reference

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Agonist-inverse agonist characterization at CB1 and CB2 cannabinoid receptors of L759633, L759656, and AM630

1 October 2017

1 reference

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The two-state model of receptor activation

1 October 2017

1 reference

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 October 2017

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Constitutive activity of cannabinoid-2 (CB2) receptors plays an essential role in the protean agonism of (+)AM1241 and L768242.

1 October 2017

1 reference

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(-)-Cannabidiol antagonizes cannabinoid receptor agonists and noradrenaline in the mouse vas deferens

23 September 2018

1 reference

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Modeling the functional effects of allosteric modulators at pharmacological receptors: an extension of the two-state model of receptor activation.

23 September 2018

1 reference

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10.1111/J.1476-5381.2011.01503.X

23 September 2018

Identifiers

DOI

1 reference

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2 February 2020

1 reference

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2 February 2020

PubMed publication ID

21615724

1 reference