SGX393 inhibits the CML mutant Bcr-AblT315I and preempts in vitro resistance when combined with nilotinib or dasatinib. (Q36535476)

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4 January 2020

title

SGX393 inhibits the CML mutant Bcr-AblT315I and preempts in vitro resistance when combined with nilotinib or dasatinib (English)

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Stephen K Burley

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author name string

Thomas O'Hare

1

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4 January 2020

Christopher A Eide

2

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Amie S Corbin

4

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Matthew J Wong

5

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Sean Buchanan

6

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4 January 2020

Kevin Holme

7

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Katayoun A Jessen

8

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Crystal Tang

9

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4 January 2020

Hal A Lewis

10

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4 January 2020

Richard D Romero

11

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Michael W Deininger

13

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language of work or name

English

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publication date

26 March 2008

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Proceedings of the National Academy of Sciences of the United States of America

4 January 2020

published in

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volume

105

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issue

14

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page(s)

5507-5512

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Crystal structure of the T315I mutant of AbI kinase

4 January 2020

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The structure of Dasatinib (BMS-354825) bound to activated ABL kinase domain elucidates its inhibitory activity against imatinib-resistant ABL mutants

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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12 December 2020

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12 December 2020

Identifiers

DOI

10.1073/PNAS.0800587105

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4 January 2020

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1 reference

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