Characterization by flow cytometry of fluorescent, selective agonist probes of the A(3) adenosine receptor. (Q36704325)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23376019%20AND%20SRC:MED&resulttype=core&format=json

23 February 2020

title

Characterization by flow cytometry of fluorescent, selective agonist probes of the A(3) adenosine receptor (English)

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23 February 2020

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6

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23 February 2020

3

Dilip K Tosh

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23 February 2020

author name string

Eszter Kozma

1

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23 February 2020

Elizabeth T Gizewski

2

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23 February 2020

Lucia Squarcialupi

4

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23 February 2020

John A Auchampach

5

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23 February 2020

language of work or name

English

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publication date

31 January 2013

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23 February 2020

published in

Biochemical Pharmacology

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23 February 2020

volume

85

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23 February 2020

issue

8

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23 February 2020

page(s)

1171-1181

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describes a project that uses

23 February 2020

1 reference

New concepts in pharmacological efficacy at 7TM receptors: IUPHAR review 2.

1 reference

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Structure-guided design of A(3) adenosine receptor-selective nucleosides: combination of 2-arylethynyl and bicyclo[3.1.0]hexane substitutions.

30 September 2017

1 reference

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Novel fluorescent antagonist as a molecular probe in A(3) adenosine receptor binding assays using flow cytometry

30 September 2017

1 reference

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Click modification in the N6 region of A3 adenosine receptor-selective carbocyclic nucleosides for dendrimeric tethering that preserves pharmacophore recognition.

30 September 2017

1 reference

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Pharmacological and therapeutic effects of A3 adenosine receptor agonists

30 September 2017

1 reference

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Novel Alexa Fluor-488 labeled antagonist of the A(2A) adenosine receptor: Application to a fluorescence polarization-based receptor binding assay

30 September 2017

1 reference

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Influence of fluorophore and linker composition on the pharmacology of fluorescent adenosine A1 receptor ligands

30 September 2017

1 reference

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2-Dialkynyl derivatives of (N)-methanocarba nucleosides: 'Clickable' A(3) adenosine receptor-selective agonists

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1 reference

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Adenosine A(3) receptor suppresses prostate cancer metastasis by inhibiting NADPH oxidase activity

30 September 2017

1 reference

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Functionalized congeners of A3 adenosine receptor-selective nucleosides containing a bicyclo[3.1.0]hexane ring system.

30 September 2017

1 reference

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30 September 2017

1 reference

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Analysis of receptor tyrosine kinase internalization using flow cytometry.

30 September 2017

1 reference

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Adenosine A(2A) receptor dynamics studied with the novel fluorescent agonist Alexa488-APEC.

30 September 2017

1 reference

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Internalization and desensitization of adenosine receptors

30 September 2017

1 reference

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The A3 adenosine receptor: an enigmatic player in cell biology

30 September 2017

1 reference

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Agonist-occupied A3 adenosine receptors exist within heterogeneous complexes in membrane microdomains of individual living cells.

30 September 2017

1 reference

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Cl-IB-MECA [2-chloro-N6-(3-iodobenzyl)adenosine-5'-N-methylcarboxamide] reduces ischemia/reperfusion injury in mice by activating the A3 adenosine receptor

30 September 2017

1 reference

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2H-NMR study and molecular dynamics simulation of the location, alignment, and mobility of pyrene in POPC bilayers

30 September 2017

1 reference

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A3 adenosine receptors in human astrocytoma cells: agonist-mediated desensitization, internalization, and down-regulation

30 September 2017

1 reference

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Inosine binds to A3 adenosine receptors and stimulates mast cell degranulation

30 September 2017

1 reference

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Induction of multiple effects on adenylyl cyclase regulation by chronic activation of the human A3 adenosine receptor

30 September 2017

1 reference

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Binding thermodynamics at A1 and A2A adenosine receptors

30 September 2017

1 reference

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

30 September 2017

1 reference

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30 September 2017

1 reference

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Control of enteric neuromuscular functions by purinergic A(3) receptors in normal rat distal colon and experimental bowel inflammation

30 September 2017

1 reference

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Highly potent and selective fluorescent antagonists of the human adenosine A₃ receptor based on the 1,2,4-triazolo[4,3-a]quinoxalin-1-one scaffold.

28 June 2018

1 reference

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New fluorescent adenosine A1-receptor agonists that allow quantification of ligand-receptor interactions in microdomains of single living cells.

5 September 2018

1 reference

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ATP release guides neutrophil chemotaxis via P2Y2 and A3 receptors.

5 September 2018

1 reference

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Activation of adenosine A3 receptors reduces ischemic brain injury in rodents.

5 September 2018

1 reference

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Adenosine inhibits tumor necrosis factor-alpha release from mouse peritoneal macrophages via A2A and A2B but not the A3 adenosine receptor

5 September 2018

1 reference

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Lysozyme effect on structural state of model membranes as revealed by pyrene excimerization studies

5 September 2018

1 reference

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The effect of inhibitors of receptor internalization on the desensitization and resensitization of three Gs-coupled receptor responses

5 September 2018

1 reference

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Adenosine receptor specificity in preconditioning of isolated rabbit cardiomyocytes: evidence of A3 receptor involvement

5 September 2018

1 reference

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Subtype-specific kinetics of inhibitory adenosine receptor internalization are determined by sensitivity to phosphorylation by G protein-coupled receptor kinases

5 September 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/23376019

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Agonist-Induced Internalization and Recycling of the Human A3 Adenosine Receptors

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/23376019

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.BCP.2013.01.021

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23376019%20AND%20SRC:MED&resulttype=core&format=json

23 February 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23376019%20AND%20SRC:MED&resulttype=core&format=json

23 February 2020

PubMed publication ID

23376019

1 reference