Structure-activity relationships of truncated D- and l-4'-thioadenosine derivatives as species-independent A3 adenosine receptor antagonists (Q36740173)

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scientific article published on 24 September 2008

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English	Structure-activity relationships of truncated D- and l-4'-thioadenosine derivatives as species-independent A3 adenosine receptor antagonists	scientific article published on 24 September 2008

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14 January 2020

Structure-activity relationships of truncated D- and l-4'-thioadenosine derivatives as species-independent A3 adenosine receptor antagonists (English)

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14 January 2020

Kenneth A. Jacobson

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14 January 2020

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Zhan-Guo Gao

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14 January 2020

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Dilip K Tosh

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14 January 2020

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Lak Shin Jeong

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14 January 2020

Hyung Ryong Moon

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Hyung Ryong Moon

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14 January 2020

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Hyuk Woo Lee

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14 January 2020

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Athena M Klutz

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14 January 2020

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Xiyan Hou

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14 January 2020

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Seung Ah Choe

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14 January 2020

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Shantanu Pal

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14 January 2020

Won Jun Choi

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14 January 2020

Hea Ok Kim

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14 January 2020

Sang Kook Lee

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14 January 2020

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24 September 2008

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14 January 2020

Journal of Medicinal Chemistry

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14 January 2020

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14 January 2020

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14 January 2020

6609-6613

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14 January 2020

Design of (N)-methanocarba adenosine 5'-uronamides as species-independent A3 receptor-selective agonists.

1 reference

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29 September 2017

Structure-activity relationships of 2-chloro-N6-substituted-4'-thioadenosine-5'-N,N-dialkyluronamides as human A3 adenosine receptor antagonists

1 reference

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29 September 2017

Discovery of a new nucleoside template for human A3 adenosine receptor ligands: D-4'-thioadenosine derivatives without 4'-hydroxymethyl group as highly potent and selective antagonists

1 reference

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29 September 2017

Docking studies of agonists and antagonists suggest an activation pathway of the A3 adenosine receptor

1 reference

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29 September 2017

Design, synthesis, and biological activity of N6-substituted-4'-thioadenosines at the human A3 adenosine receptor

1 reference

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29 September 2017

Adenosine receptors as therapeutic targets

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29 September 2017

Structure-activity relationships of 2-chloro-N6-substituted-4'-thioadenosine-5'-uronamides as highly potent and selective agonists at the human A3 adenosine receptor

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A novel adenosine analog, thio-Cl-IB-MECA, induces G0/G1 cell cycle arrest and apoptosis in human promyelocytic leukemia HL-60 cells

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Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine ligands, new tools to characterize A3 adenosine receptors in human tumor cell lines

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2-Substituted adenosine derivatives: affinity and efficacy at four subtypes of human adenosine receptors

1 reference

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29 September 2017

Modulation of adenosine receptor affinity and intrinsic efficacy in adenine nucleosides substituted at the 2-position

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29 September 2017

N6-substituted D-4'-thioadenosine-5'-methyluronamides: potent and selective agonists at the human A3 adenosine receptor

1 reference

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29 September 2017

N6-Substituted adenosine derivatives: selectivity, efficacy, and species differences at A3 adenosine receptors

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29 September 2017

Adenosine receptors and their ligands.

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Anilide derivatives of an 8-phenylxanthine carboxylic congener are highly potent and selective antagonists at human A(2B) adenosine receptors

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A(3) adenosine receptor ligands: history and perspectives

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The role of receptor structure in determining adenosine receptor activity

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Biochemical methods for detection and measurement of cyclic AMP and adenylyl cyclase activity.

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2-Substitution of N6-benzyladenosine-5'-uronamides enhances selectivity for A3 adenosine receptors

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Structure-activity relationships of 9-alkyladenine and ribose-modified adenosine derivatives at rat A3 adenosine receptors

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Comparative pharmacology of human adenosine receptor subtypes - characterization of stably transfected receptors in CHO cells.

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Structural determinants of A(3) adenosine receptor activation: nucleoside ligands at the agonist/antagonist boundary

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The antitumor effect of LJ-529, a novel agonist to A3 adenosine receptor, in both estrogen receptor-positive and estrogen receptor-negative human breast cancers

1 reference

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Stereoselective functionalization of the 1'-position of 4'-thionucleosides

1 reference

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Identifiers

10.1021/JM8008647

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14 January 2020

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14 January 2020

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14 January 2020

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