Bisthiazolidines: A Substrate-Mimicking Scaffold as an Inhibitor of the NDM-1 Carbapenemase (Q37340068)

19 August 2017

Bisthiazolidines: A Substrate-Mimicking Scaffold as an Inhibitor of the NDM-1 Carbapenemase (English)

1 reference

19 August 2017

Christopher J. Schofield

8

1 reference

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31 May 2020

Philip Hinchliffe

5

1 reference

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31 May 2020

Jürgen Brem

7

1 reference

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31 May 2020

Graciela Mahler

9

1 reference

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31 May 2020

Leticia I Llarrull

11

1 reference

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31 May 2020

author name string

Mariano M González

1

1 reference

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31 May 2020

Magda Kosmopoulou

2

1 reference

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31 May 2020

Maria F Mojica

3

1 reference

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31 May 2020

Valerie Castillo

4

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31 May 2020

Ilaria Pettinati

6

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31 May 2020

James Spencer

12

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31 May 2020

Alejandro J Vila

13

1 reference

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31 May 2020

Robert A Bonomo

10

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31 May 2020

publication date

20 July 2015

1 reference

19 August 2017

ACS Infectious Diseases

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31 May 2020

volume

1

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31 May 2020

issue

11

1 reference

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31 May 2020

page(s)

544-554

1 reference

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Exploring the Role of Residue 228 in Substrate and Inhibitor Recognition by VIM Metallo-β-lactamases

31 May 2020

cites work

1 reference

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Approved Drugs Containing Thiols as Inhibitors of Metallo-β-lactamases: Strategy To Combat Multidrug-Resistant Bacteria

6 September 2017

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Rhodanine hydrolysis leads to potent thioenolate mediated metallo-β-lactamase inhibition

6 September 2017

1 reference

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Structural and mechanistic insights into NDM-1 catalyzed hydrolysis of cephalosporins

6 September 2017

1 reference

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Molecular mechanisms of substrate recognition and specificity of New Delhi metallo-β-lactamase

6 September 2017

1 reference

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Aspergillomarasmine A overcomes metallo-β-lactamase antibiotic resistance

6 September 2017

1 reference

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Discovering Echinococcus granulosus thioredoxin glutathione reductase inhibitors through site-specific dynamic combinatorial chemistry.

6 September 2017

1 reference

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Clinical epidemiology of the global expansion of Klebsiella pneumoniae carbapenemases

6 September 2017

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Antibiotic resistance in Zn(II)-deficient environments: metallo-β-lactamase activation in the periplasm.

6 September 2017

1 reference

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The glyoxalase pathway: the first hundred years... and beyond

6 September 2017

1 reference

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Carbapenem-resistant Enterobacteriaceae: a review of treatment and outcomes

6 September 2017

1 reference

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New Delhi metallo-β-lactamase: structural insights into β-lactam recognition and inhibition

6 September 2017

1 reference

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Towards automated crystallographic structure refinement with phenix.refine

6 September 2017

1 reference

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Structure of Apo- and Monometalated Forms of NDM-1—A Highly Potent Carbapenem-Hydrolyzing Metallo-β-Lactamase

6 September 2017

1 reference

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Crystal structure of New Delhi metallo-β-lactamase reveals molecular basis for antibiotic resistance

6 September 2017

1 reference

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Increasing prevalence and dissemination of NDM-1 metallo-β-lactamase in India: data from the SMART study (2009)

6 September 2017

1 reference

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A structural view of the antibiotic degradation enzyme NDM-1 from a superbug

6 September 2017

1 reference

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Status report on carbapenemases: challenges and prospects

6 September 2017

1 reference

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Crystal structure of NDM-1 reveals a common β-lactam hydrolysis mechanism

6 September 2017

1 reference

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Dissemination of NDM-1 positive bacteria in the New Delhi environment and its implications for human health: an environmental point prevalence study.

6 September 2017

1 reference

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An introduction to data reduction: space-group determination, scaling and intensity statistics

6 September 2017

1 reference

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Overview of the CCP4 suite and current developments

6 September 2017

1 reference

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Alarming β-lactamase-mediated resistance in multidrug-resistant Enterobacteriaceae

6 September 2017

1 reference

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Emergence of a new antibiotic resistance mechanism in India, Pakistan, and the UK: a molecular, biological, and epidemiological study

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5064445

Features and development of Coot

6 September 2017

1 reference

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Integration, scaling, space-group assignment and post-refinement

6 September 2017

1 reference

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MolProbity: all-atom structure validation for macromolecular crystallography

6 September 2017

1 reference

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Characterization of a new metallo-beta-lactamase gene, bla(NDM-1), and a novel erythromycin esterase gene carried on a unique genetic structure in Klebsiella pneumoniae sequence type 14 from India

6 September 2017

1 reference

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Microwave assisted tandem reactions for the synthesis of 2-hydrazolyl-4-thiazolidinones

6 September 2017

1 reference

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Phasercrystallographic software

6 September 2017

1 reference

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Trapping and characterization of a reaction intermediate in carbapenem hydrolysis by B. cereus metallo-beta-lactamase

6 September 2017

1 reference

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Dynamic combinatorial mass spectrometry leads to metallo-beta-lactamase inhibitors

6 September 2017

1 reference

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Global challenge of multidrug-resistant Acinetobacter baumannii

6 September 2017

1 reference

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Metallo-beta-lactamases (classification, activity, genetic organization, structure, zinc coordination) and their superfamily

6 September 2017

1 reference

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A versatile ligation-independent cloning method suitable for high-throughput expression screening applications

6 September 2017

1 reference

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Metallo-beta-lactamases: novel weaponry for antibiotic resistance in bacteria

6 September 2017

1 reference

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Scaling and assessment of data quality

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5064445

Bacterial resistance to beta-lactam antibiotics: compelling opportunism, compelling opportunity

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5064445

Secondary-structure matching (SSM), a new tool for fast protein structure alignment in three dimensions

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5064445

Reliable high-throughput functional screening with 3-FABS.

6 September 2017

1 reference

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The 1.5-A structure of Chryseobacterium meningosepticum zinc beta-lactamase in complex with the inhibitor, D-captopril

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5064445

Tobacco etch virus protease: mechanism of autolysis and rational design of stable mutants with wild-type catalytic proficiency

6 September 2017

1 reference

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Succinic acids as potent inhibitors of plasmid-borne IMP-1 metallo-beta-lactamase

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5064445

Standard numbering scheme for class B beta-lactamases

6 September 2017

1 reference

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On the mechanism of the metallo-beta-lactamase from Bacteroides fragilis

6 September 2017

1 reference

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Gamma-lactam analogues of beta-lactam antibiotics

6 September 2017

1 reference

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Crystallization and preliminary X-ray crystallographic analysis of the [NiFe]-hydrogenase maturation factor HypF1 from Ralstonia eutropha H16

6 September 2017

1 reference

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Monitoring conformational changes in the NDM-1 metallo-β-lactamase by 19F NMR spectroscopy

14 September 2017

1 reference

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Interaction of the C-terminal domains of sendai virus N and P proteins: comparison of polymerase-nucleocapsid interactions within the paramyxovirus family

28 September 2017

1 reference

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Real-time monitoring of New Delhi metallo-β-lactamase activity in living bacterial cells by 1H NMR spectroscopy

26 June 2018

1 reference

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Activity of carbapenems with ME1071 (disodium 2,3-diethylmaleate) against Enterobacteriaceae and Acinetobacter spp. with carbapenemases, including NDM enzymes

2 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5064445

A metallo-beta-lactamase enzyme in action: crystal structures of the monozinc carbapenemase CphA and its complex with biapenem

2 September 2018

1 reference

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Structural determinants of substrate binding to Bacillus cereus metallo-beta-lactamase

2 September 2018

1 reference

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Thiomandelic acid, a broad spectrum inhibitor of zinc beta-lactamases: kinetic and spectroscopic studies

2 September 2018

1 reference

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Outer membrane permeability of Acinetobacter calcoaceticus and its implication in antibiotic resistance

2 September 2018

1 reference

12 December 2020

Diaryl-substituted azolylthioacetamides: Inhibitor discovery of New Delhi metallo-β-lactamase-1 (NDM-1)

1 reference

12 December 2020

Mechanistic and spectroscopic studies of metallo-β-lactamase NDM-1

1 reference

12 December 2020

A minimalistic approach to identify substrate binding features in B1 Metallo-beta-lactamases

1 reference

12 December 2020

10.1021/ACSINFECDIS.5B00046

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27623409%20AND%20SRC:MED&resulttype=core&format=json

31 May 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27623409%20AND%20SRC:MED&resulttype=core&format=json

31 May 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:27623409%20AND%20SRC:MED&resulttype=core&format=json