Development of a fluorescence polarization based assay for histone deacetylase ligand discovery (Q38787596)

6 September 2017

Development of a fluorescence polarization based assay for histone deacetylase ligand discovery (English)

1 reference

6 September 2017

3

Dyann F Wirth

1 reference

6 September 2017

1

Ralph Mazitschek

0 references

Jon Clardy

series ordinal

4

object named as

Jon Clardy

1 reference

6 September 2017

Ralph Mazitschek

1

1 reference

PMCID

2408937

6 September 2017

Vishal Patel

series ordinal

2

1 reference

PMCID

2408937

6 September 2017

language of work or name

English

0 references

publication date

7 April 2008

1 reference

Bioorganic & Medicinal Chemistry Letters

6 September 2017

1 reference

6 September 2017

18

1 reference

6 September 2017

2809-2812

1 reference

6 September 2017

9

1 reference

Unraveling the hidden catalytic activity of vertebrate class IIa histone deacetylases

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

Dimethyl sulfoxide to vorinostat: development of this histone deacetylase inhibitor as an anticancer drug

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

Histone deacetylase inhibitors and the promise of epigenetic (and more) treatments for cancer

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

Epigenetic and chromatin modifiers as targeted therapy of hematologic malignancies

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

The silencing protein SIR2 and its homologs are NAD-dependent protein deacetylases

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

Transcriptional silencing and longevity protein Sir2 is an NAD-dependent histone deacetylase

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

A class of hybrid polar inducers of transformed cell differentiation inhibits histone deacetylases.

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

A mammalian histone deacetylase related to the yeast transcriptional regulator Rpd3p

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

Changing patterns of histone acetylation and RNA synthesis in regeneration of the liver

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

A non-isotopic assay for histone deacetylase activity

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

Effect of DNase I on histone acetyltransferase and deacetylase enzyme activities in friend cell nuclei: Evidence for a putative inhibitor of the deacetylase enzymes in transcriptionally active chromatin

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

Suberoylanilide hydroxamic acid (SAHA) overcomes multidrug resistance and induces cell death in P-glycoprotein-expressing cells

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

The histone deacetylase inhibitor MS-275 promotes differentiation or apoptosis in human leukemia cells through a process regulated by generation of reactive oxygen species and induction of p21CIP1/WAF1 1.

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

1 Equilibrium and kinetic inhibition assays based upon fluorescence polarization

23 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

An exact correction to the "Cheng-Prusoff" correction.

23 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

Molecular evolution of the histone deacetylase family: functional implications of phylogenetic analysis.

23 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

Improved fluorogenic histone deacetylase assay for high-throughput-screening applications

31 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

A fluorogenic histone deacetylase assay well suited for high-throughput activity screening

31 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

Fluorescence anisotropy applied to biomolecular interactions.

31 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2408937

Fluorescence polarization — a new tool for cell and molecular biology

31 August 2018

1 reference

12 December 2020

Amide Analogues of Trichostatin A as Inhibitors of Histone Deacetylase and Inducers of Terminal Cell Differentiation

1 reference

12 December 2020

Enzymatic deacetylation of histone

1 reference

12 December 2020

Acetylation of histones by pigeon liver enzymes

1 reference

12 December 2020

Factors affecting the substrate specificity of histone deacetylases

1 reference

12 December 2020

10.1016/J.BMCL.2008.04.007

Identifiers

DOI

1 reference

6 September 2017

1 reference

6 September 2017

1 reference

PMCID

2408937