Activation of Hsp90 Enzymatic Activity and Conformational Dynamics through Rationally Designed Allosteric Ligands. (Q38842676)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26286886%20AND%20SRC:MED&resulttype=core&format=json

22 February 2020

title

Activation of Hsp90 Enzymatic Activity and Conformational Dynamics through Rationally Designed Allosteric Ligands (English)

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22 February 2020

1

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Anna Bernardi

18

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22 February 2020

Giorgio Colombo

19

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22 February 2020

Marzia Pennati

5

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22 February 2020

Laura Morelli

7

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22 February 2020

Abbey D Zuehlke

9

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Marco Rusnati

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22 February 2020

Nadia Zaffaroni

16

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22 February 2020

15

Len Neckers

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22 February 2020

2

Jiahui Tao

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4

Elisabetta Moroni

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22 February 2020

13

Kristin Beebe

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22 February 2020

author name string

Gerolamo Vettoretti

3

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22 February 2020

Alessia Lopergolo

6

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22 February 2020

Antonella Bugatti

8

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22 February 2020

Mike Moses

10

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22 February 2020

Thomas Prince

11

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Toshiki Kijima

12

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22 February 2020

David A Agard

17

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22 February 2020

language of work or name

English

0 references

publication date

18 August 2015

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Chemistry—A European Journal

22 February 2020

published in

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volume

21

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issue

39

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22 February 2020

page(s)

13598-13608

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GROMACS 4: Algorithms for Highly Efficient, Load-Balanced, and Scalable Molecular Simulation

22 February 2020

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Posttranslational modification and conformational state of heat shock protein 90 differentially affect binding of chemically diverse small molecule inhibitors

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30 June 2018

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30 June 2018

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30 June 2018

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30 June 2018

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30 June 2018

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30 June 2018

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30 June 2018

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ATP binding and hydrolysis are essential to the function of the Hsp90 molecular chaperone in vivo

30 June 2018

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22 August 2018

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Dissection of the ATP-induced conformational cycle of the molecular chaperone Hsp90.

22 August 2018

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Survivin is highly expressed and promotes cell survival in malignant peritoneal mesothelioma.

22 August 2018

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22 August 2018

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21 January 2018

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21 January 2018

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Artificial Accelerators of the Molecular Chaperone Hsp90 Facilitate Rate-Limiting Conformational Transitions

4 November 2018

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Synthesis of potential allosteric modulators of Hsp90 by chemical glycosylation of Eupomatenoid-6

21 January 2018

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Asymmetric Activation of the Hsp90 Dimer by Its Cochaperone Aha1

2 December 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/26286886

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Hsp90 regulation of endothelial nitric oxide synthase contributes to vascular control in portal hypertension

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/26286886

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1002/CHEM.201502211

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26286886%20AND%20SRC:MED&resulttype=core&format=json

22 February 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26286886%20AND%20SRC:MED&resulttype=core&format=json

22 February 2020

PubMed publication ID

26286886

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26286886%20AND%20SRC:MED&resulttype=core&format=json