Internalization of CCR4 and inhibition of chemotaxis by K777, a potent and selective CCR4 antagonist (Q39141759)

9 September 2017

title

Internalization of CCR4 and inhibition of chemotaxis by K777, a potent and selective CCR4 antagonist (English)

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9 September 2017

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Takashi Sato

1

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9 September 2017

Miho Iwase

2

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9 September 2017

Motoki Miyama

3

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9 September 2017

Masato Komai

4

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9 September 2017

Etsuo Ohshima

5

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9 September 2017

Akira Asai

6

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9 September 2017

Hiroshi Yano

7

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9 September 2017

Ichiro Miki

8

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9 September 2017

publication date

5 June 2013

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9 September 2017

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9 September 2017

volume

91

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9 September 2017

issue

5-6

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9 September 2017

page(s)

305-313

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GPCR expression in tissues and cells: are the optimal receptors being used as drug targets?

9 September 2017

cites work

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New insights into the regulation of cAMP synthesis beyond GPCR/G protein activation: implications in cardiovascular regulation.

21 January 2018

1 reference

GPCR agonists and antagonists in the clinic

21 January 2018

1 reference

Biochemical mechanisms of drug action: what does it take for success?

21 January 2018

1 reference

Uncovering molecular mechanisms involved in activation of G protein-coupled receptors

21 January 2018

1 reference

Taking the time to study competitive antagonism

21 January 2018

1 reference

Positive allosteric modulators of metabotropic glutamate 1 receptor: characterization, mechanism of action, and binding site

21 January 2018

1 reference

Allosteric modulation of G protein-coupled receptors.

21 January 2018

1 reference

Chemokines--chemotactic cytokines that mediate inflammation

21 January 2018

1 reference

Chemokines, chemokine receptors and allergy

21 January 2018

1 reference

T-cell subsets: recruiting the right kind of help

21 January 2018

1 reference

Solution structure and basis for functional activity of stromal cell-derived factor-1; dissociation of CXCR4 activation from binding and inhibition of HIV-1.

21 January 2018

1 reference

N-terminal peptides of stromal cell-derived factor-1 with CXC chemokine receptor 4 agonist and antagonist activities

21 January 2018

1 reference

The T cell-directed CC chemokine TARC is a highly specific biological ligand for CC chemokine receptor 4

21 January 2018

1 reference

Macrophage-derived chemokine is a functional ligand for the CC chemokine receptor 4

21 January 2018

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Unique chemotactic response profile and specific expression of chemokine receptors CCR4 and CCR8 by CD4(+)CD25(+) regulatory T cells

21 January 2018

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Regulatory T cells accumulate in the lung allergic inflammation and efficiently suppress T-cell proliferation but not Th2 cytokine production

21 January 2018

1 reference

Inducible expression of a Th2-type CC chemokine thymus- and activation-regulated chemokine by human bronchial epithelial cells

21 January 2018

1 reference

The C-C chemokine receptors CCR4 and CCR8 identify airway T cells of allergen-challenged atopic asthmatics

21 January 2018

1 reference

Demonstration of TARC and CCR4 mRNA expression and distribution using in situ RT-PCR in the lesional skin of atopic dermatitis

21 January 2018

1 reference

CCR4 in human allergen-induced late responses in the skin and lung

21 January 2018

1 reference

Chemokine receptor antagonists: Part 1.

21 January 2018

1 reference

Optimization of 2-aminothiazole derivatives as CCR4 antagonists

21 January 2018

1 reference

Discovery and SAR of trisubstituted thiazolidinones as CCR4 antagonists

21 January 2018

1 reference

Discovery of potent CCR4 antagonists: Synthesis and structure-activity relationship study of 2,4-diaminoquinazolines

21 January 2018

1 reference

Core exploration in optimization of chemokine receptor CCR4 antagonists

21 January 2018

1 reference

Inhibitory effect of the new orally active CCR4 antagonist K327 on CCR4+CD4+ T cell migration into the lung of mice with ovalbumin-induced lung allergic inflammation

21 January 2018

1 reference

Human cutaneous T cell lymphoma and leukemia cell lines produce and respond to T cell growth factor

21 January 2018

1 reference

Establishment and characterization of a new leukaemic T-cell line (Peer) with an unusual phenotype.

21 January 2018

1 reference

The noncompetitive antagonism of histamine H1 receptors expressed in Chinese hamster ovary cells by olopatadine hydrochloride: its potency and molecular mechanism

21 January 2018

1 reference

Dominance of CCL22 over CCL17 in induction of chemokine receptor CCR4 desensitization and internalization on human Th2 cells

21 January 2018

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Functional Selectivity and Classical Concepts of Quantitative Pharmacology

21 January 2018

1 reference

21 January 2018

Identifiers

DOI

10.1159/000350390

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9 September 2017

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