Expression and functional properties of canine, rat, and murine histamine H₄ receptors in Sf9 insect cells. (Q39584467)

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23 January 2020

title

Expression and functional properties of canine, rat, and murine histamine H₄ receptors in Sf9 insect cells (English)

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23 January 2020

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23 January 2020

author name string

David Schnell

1

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23 January 2020

Irena Brunskole

2

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23 January 2020

Katerina Ladova

3

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23 January 2020

Patrick Igel

5

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23 January 2020

Stefan Dove

6

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23 January 2020

Armin Buschauer

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Roland Seifert

8

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publication date

27 February 2011

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Naunyn-Schmiedeberg's Archives of Pharmacology

23 January 2020

published in

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23 January 2020

volume

383

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23 January 2020

issue

5

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23 January 2020

page(s)

457-470

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Definition and antagonism of histamine H 2 -receptors

23 January 2020

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Histamine induces cytoskeletal changes in human eosinophils via the H4 receptor

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Antiinflammatory and antinociceptive effects of the selective histamine H4-receptor antagonists JNJ7777120 and VUF6002 in a rat model of carrageenan-induced acute inflammation

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The histamine H4 receptor mediates inflammation and pruritus in Th2-dependent dermal inflammation

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Cationic-amphiphilic arpromidine-derived guanidines and a histamine trifluoromethyl-toluidide derivative may activate pertussis toxin-sensitive G-proteins by a receptor-independent mechanism

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Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist

21 January 2018

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Phenylalanine 169 in the second extracellular loop of the human histamine H4 receptor is responsible for the difference in agonist binding between human and mouse H4 receptors

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Histamine H4 receptor mediates eosinophil chemotaxis with cell shape change and adhesion molecule upregulation

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Histamine 4 receptor activation induces recruitment of FoxP3+ T cells and inhibits allergic asthma in a murine model.

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Does the histamine H4 receptor have a pro- or anti-inflammatory role in murine bronchial asthma?

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Identification of a histamine H4 receptor on human eosinophils--role in eosinophil chemotaxis

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Constitutive activity and ligand selectivity of human, guinea pig, rat, and canine histamine H2 receptors

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GTPase-activating proteins for heterotrimeric G proteins: regulators of G protein signaling (RGS) and RGS-like proteins

21 January 2018

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Histamine H4 receptor antagonism reduces hapten-induced scratching behaviour but not inflammation.

21 January 2018

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The histamine H receptor as a new target for treatment of canine inflammatory skin diseases.

21 January 2018

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Histamine H(4) receptor-RGS fusion proteins expressed in Sf9 insect cells: a sensitive and reliable approach for the functional characterization of histamine H(4) receptor ligands.

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21 January 2018

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Identifiers

DOI

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23 January 2020

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