Bromodomains: are readers right for epigenetic therapy? (Q39734340)

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20 March 2020

editorial

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title

Bromodomains: are readers right for epigenetic therapy? (English)

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20 March 2020

1

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20 March 2020

author name string

Stuart J Conway

series ordinal

1

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14 September 2017

9 August 2012

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24900532%20AND%20SRC:MED&resulttype=core&format=json

ACS Medicinal Chemistry Letters

20 March 2020

published in

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20 March 2020

volume

3

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20 March 2020

issue

9

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20 March 2020

page(s)

691-694

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The bromodomain interaction module

20 March 2020

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

Down-regulation of NF-κB transcriptional activity in HIV-associated kidney disease by BRD4 inhibition

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

Epigenetic protein families: a new frontier for drug discovery

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

Identification of a novel series of BET family bromodomain inhibitors: binding mode and profile of I-BET151 (GSK1210151A)

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

Fragment-based discovery of bromodomain inhibitors part 2: optimization of phenylisoxazole sulfonamides

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

Inhibition of BET recruitment to chromatin as an effective treatment for MLL-fusion leukaemia

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

BET bromodomain inhibition as a therapeutic strategy to target c-Myc

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

3,5-dimethylisoxazoles act as acetyl-lysine-mimetic bromodomain ligands

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

RNAi screen identifies Brd4 as a therapeutic target in acute myeloid leukaemia

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

Suppression of inflammation by a synthetic histone mimic

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

Selective inhibition of BET bromodomains

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

Selective small molecules blocking HIV-1 Tat and coactivator PCAF association

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

Acetylation: a regulatory modification to rival phosphorylation?

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

The bromodomain: a conserved sequence found in human, Drosophila and yeast proteins

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

Druggability analysis and structural classification of bromodomain acetyl-lysine binding sites

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025779

15 June 2018

Identifiers

DOI

10.1021/ML300221T

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24900532%20AND%20SRC:MED&resulttype=core&format=json

20 March 2020

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24900532%20AND%20SRC:MED&resulttype=core&format=json

20 March 2020

PubMed publication ID

24900532

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24900532%20AND%20SRC:MED&resulttype=core&format=json