Rational design of RAR-selective ligands revealed by RARbeta crystal structure (Q40104851)

17 September 2017

Rational design of RAR-selective ligands revealed by RARbeta crystal structure (English)

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17 September 2017

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17 September 2017

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17 September 2017

Angel R de Lera

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Pierre Germain

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object named as

Pierre Germain

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17 September 2017

Sabrina Kammerer

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17 September 2017

Efrén Pérez

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Carole Peluso-Iltis

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17 September 2017

David Tortolani

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F Christopher Zusi

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17 September 2017

John Starrett

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17 September 2017

Philippe Lapointe

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17 September 2017

Jean-Paul Daris

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17 September 2017

Anne Marinier

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17 September 2017

1 September 2004

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877-882

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Principles for modulation of the nuclear receptor superfamily

17 September 2017

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

Estrogen receptor-alpha directs ordered, cyclical, and combinatorial recruitment of cofactors on a natural target promoter

22 September 2017

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

The promise of retinoids to fight against cancer.

22 September 2017

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

Retinoids and their receptors in cancer development and chemoprevention

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

Epigenetic downregulation of the retinoic acid receptor-beta2 gene in breast cancer.

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

Nuclear receptor ligand-binding domains: three-dimensional structures, molecular interactions and pharmacological implications

22 September 2017

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

Structural basis for isotype selectivity of the human retinoic acid nuclear receptor

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

Crystal structure of a heterodimeric complex of RAR and RXR ligand-binding domains

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

Enantiomer discrimination illustrated by high-resolution crystal structures of the human nuclear receptor hRARgamma

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

Structural basis for engineering of retinoic acid receptor isotype-selective agonists and antagonists

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

Conformational adaptation of agonists to the human nuclear receptor RAR gamma

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

A mutation mimicking ligand-induced conformational change yields a constitutive RXR that senses allosteric effects in heterodimers

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

RARs and RXRs: evidence for two autonomous transactivation functions (AF-1 and AF-2) and heterodimerization in vivo

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

RAR-specific agonist/antagonists which dissociate transactivation and AP1 transrepression inhibit anchorage-independent cell proliferation.

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

Crystal structure of the RAR-gamma ligand-binding domain bound to all-trans retinoic acid

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

Co-regulator recruitment and the mechanism of retinoic acid receptor synergy

22 September 2017

1 reference

Crossref

https://api.crossref.org/works/10.1038%2FSJ.EMBOR.7400235

Endogenous reactivation of the RARbeta2 tumor suppressor gene epigenetically silenced in breast cancer.

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1299136

20 August 2018

Identifiers

DOI

10.1038/SJ.EMBOR.7400235

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17 September 2017

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17 September 2017

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