Exploring the potential of boronic acids as inhibitors of OXA-24/40 β-lactamase (Q40402495)

23 May 2018

title

Exploring the potential of boronic acids as inhibitors of OXA-24/40 β-lactamase (English)

1 reference

23 May 2018

1 reference

boronic acids

15 July 2023

4

Robert A Bonomo

1 reference

23 May 2018

0 references

Josephine P Werner

1

1 reference

23 May 2018

Joshua M Mitchell

series ordinal

2

1 reference

23 May 2018

Magdalena A Taracila

series ordinal

3

1 reference

23 May 2018

Rachel A Powers

series ordinal

5

1 reference

23 May 2018

publication date

23 February 2017

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23 May 2018

published in

Protein Science

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23 May 2018

volume

26

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23 May 2018

page(s)

515-526

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23 May 2018

issue

3

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23 May 2018

The structure of a doripenem-bound OXA-51 class D β-lactamase variant with enhanced carbapenemase activity

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Structural Basis for Enhancement of Carbapenemase Activity in the OXA-51 Family of Class D β-Lactamases

17 June 2018

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Discovery of a Cyclic Boronic Acid β-Lactamase Inhibitor (RPX7009) with Utility vs Class A Serine Carbapenemases

17 June 2018

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17 June 2018

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Targeting Class A and C Serine β-Lactamases with a Broad-Spectrum Boronic Acid Derivative

17 June 2018

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Crystal Structure of Carbapenemase OXA-58 from Acinetobacter baumannii

17 June 2018

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17 June 2018

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17 June 2018

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17 June 2018

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17 June 2018

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17 June 2018

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17 June 2018

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17 June 2018

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17 June 2018

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Structures of the Class D Carbapenemase OXA-24 from Acinetobacter baumannii in Complex with Doripenem

17 June 2018

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17 June 2018

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4,7-Dichloro benzothien-2-yl sulfonylaminomethyl boronic acid: first boronic acid-derived beta-lactamase inhibitor with class A, C, and D activity

17 June 2018

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Three decades of beta-lactamase inhibitors

17 June 2018

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17 June 2018

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Updated functional classification of beta-lactamases

17 June 2018

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Diversity, epidemiology, and genetics of class D beta-lactamases

17 June 2018

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In vitro activity of NXL104 in combination with beta-lactams against Klebsiella pneumoniae isolates producing KPC carbapenemases

17 June 2018

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Crystal structure of the OXA-48 beta-lactamase reveals mechanistic diversity among class D carbapenemases

17 June 2018

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17 June 2018

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17 June 2018

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17 June 2018

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17 June 2018

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17 June 2018

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17 June 2018

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Inhibition of class D beta-lactamases by acyl phosphates and phosphonates

17 June 2018

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Identification of a new allelic variant of the Acinetobacter baumannii cephalosporinase, ADC-7 beta-lactamase: defining a unique family of class C enzymes

17 June 2018

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Refinement of macromolecular structures by the maximum-likelihood method

17 June 2018

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Nanomolar inhibitors of AmpC beta-lactamase

17 June 2018

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Structure-based approach for binding site identification on AmpC beta-lactamase

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5326569

17 June 2018

b-Lactamase inhibitors

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Structure-based design guides the improved efficacy of deacylation transition state analogue inhibitors of TEM-1 beta-Lactamase(,)

17 June 2018

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Cloning, nucleotide sequencing, and analysis of the gene encoding an AmpC beta-lactamase in Acinetobacter baumannii

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5326569

Three-dimensional structure of AmpC beta-lactamase from Escherichia coli bound to a transition-state analogue: possible implications for the oxyanion hypothesis and for inhibitor design

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5326569

pi-Stacking interactions. Alive and well in proteins

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5326569

The inhibition of class C beta-lactamases by boronic acids

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5326569

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5326569

Aromatic-aromatic interaction: a mechanism of protein structure stabilization

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5326569

ARI 1: beta-lactamase-mediated imipenem resistance in Acinetobacter baumannii.

17 June 2018

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Synthesis and SAR of novel benzoxaboroles as a new class of β-lactamase inhibitors

20 August 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/27997706

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Structure-based design of a potent transition state analogue for TEM-1 beta-lactamase

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/27997706

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Aromatic-aromatic interactions in proteins: beyond the dimer

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/27997706

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1002/PRO.3100

1 reference

23 May 2018

PMCID

5326569

1 reference

23 May 2018

PubMed ID

27997706

1 reference

23 May 2018