Constitutive internalization of constitutively active agiotensin II AT(1A) receptor mutants is blocked by inverse agonists (Q40765666)

23 September 2017

title

Constitutive internalization of constitutively active agiotensin II AT(1A) receptor mutants is blocked by inverse agonists (English)

1 reference

23 September 2017

author

Stéphanie Miserey-Lenkei

series ordinal

1

object named as

Stéphanie Miserey-Lenkei

1 reference

23 September 2017

4

Pierre Corvol

1 reference

23 September 2017

Charles Parnot

2

1 reference

23 September 2017

Sabine Bardin

series ordinal

3

1 reference

23 September 2017

Eric Clauser

series ordinal

5

1 reference

23 September 2017

language of work or name

English

0 references

publication date

29 November 2001

1 reference

Journal of Biological Chemistry

23 September 2017

published in

1 reference

23 September 2017

volume

277

1 reference

23 September 2017

issue

8

1 reference

23 September 2017

page(s)

5891-5901

1 reference

The Sequence of the Human Genome

23 September 2017

cites work

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Isolation of a cDNA encoding the vascular type-1 angiotensin II receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Phosphorylation of the type 1A angiotensin II receptor by G protein-coupled receptor kinases and protein kinase C

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Intracellular trafficking of angiotensin II and its AT1 and AT2 receptors: evidence for selective sorting of receptor and ligand

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Role of carboxyl tail of the rat angiotensin II type 1A receptor in agonist-induced internalization of the receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Short-term desensitization of the angiotensin II receptor of bovine adrenal glomerulosa cells corresponds to a shift from a high to a low affinity state

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Mutation of Asn111 in the third transmembrane domain of the AT1A angiotensin II receptor induces its constitutive activation.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

The conformational change responsible for AT1 receptor activation is dependent upon two juxtaposed asparagine residues on transmembrane helices III and VII.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Systematic identification of mutations that constitutively activate the angiotensin II type 1A receptor by screening a randomly mutated cDNA library with an original pharmacological bioassay

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Replacement of insulin receptor tyrosine residues 1162 and 1163 compromises insulin-stimulated kinase activity and uptake of 2-deoxyglucose

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Synthetic cDNA encoding the rat AT1a receptor: a useful tool for structure-function relationship analysis

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Rapid changes of mitochondrial Ca2+ revealed by specifically targeted recombinant aequorin

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

A highly sensitive quantitative cytosensor technique for the identification of receptor ligands in tissue extracts

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Constitutive activation of muscarinic receptors by the G-protein Gq.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Regulated endocytosis of G-protein-coupled receptors by a biochemically and functionally distinct subpopulation of clathrin-coated pits

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Pharmacological chaperones rescue cell-surface expression and function of misfolded V2 vasopressin receptor mutants

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Cellular distribution of constitutively active mutant parathyroid hormone (PTH)/PTH-related protein receptors and regulation of cyclic adenosine 3',5'-monophosphate signaling by beta-arrestin2.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Mechanisms governing the activation and trafficking of yeast G protein-coupled receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Mutations that induce constitutive activation and mutations that impair signal transduction modulate the basal and/or agonist-stimulated internalization of the Lutropin/Choriogonadotropin receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Effect of activating and inactivating mutations on the phosphorylation and trafficking of the human lutropin/choriogonadotropin receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

A constitutively active mutant beta 2-adrenergic receptor is constitutively desensitized and phosphorylated

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

A constitutively active mutant thyrotropin-releasing hormone receptor is chronically down-regulated in pituitary cells: evidence using chlordiazepoxide as a negative antagonist

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Up-regulation of the levels of expression and function of a constitutively active mutant of the hamster alpha1B-adrenoceptor by ligands that act as inverse agonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Inverse agonism of histamine H2 antagonist accounts for upregulation of spontaneously active histamine H2 receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Up-regulation of a constitutively active form of the beta2-adrenoceptor by sustained treatment with inverse agonists but not antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Functional consequences of constitutively active alpha2A-adrenergic receptor expression in 3T3F442A preadipocytes and adipocytes.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Structural instability of a constitutively active G protein-coupled receptor. Agonist-independent activation due to conformational flexibility

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Ligand-induced overexpression of a constitutively active beta2-adrenergic receptor: pharmacological creation of a phenotype in transgenic mice

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Role of the thrombin receptor's cytoplasmic tail in intracellular trafficking. Distinct determinants for agonist-triggered versus tonic internalization and intracellular localization

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Visualization of G protein-coupled receptor trafficking with the aid of the green fluorescent protein. Endocytosis and recycling of cholecystokinin receptor type A

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Constitutive arrestin-mediated desensitization of a human vasopressin receptor mutant associated with nephrogenic diabetes insipidus

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Agonist-induced phosphorylation of the angiotensin II (AT(1A)) receptor requires generation of a conformation that is distinct from the inositol phosphate-signaling state

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Removal of phosphorylation sites from the β2-adrenergic receptor delays onset of agonist-promoted desensitization

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Inverse agonism and the regulation of receptor number

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Stable expression of a truncated AT1A receptor in CHO-K1 cells. The carboxyl-terminal region directs agonist-induced internalization but not receptor signaling or desensitization.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

Mutation of Asp74 of the rat angiotensin II receptor confers changes in antagonist affinities and abolishes G-protein coupling.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M108398200

21 January 2018

Identifiers

DOI

10.1074/JBC.M108398200

1 reference

23 September 2017

1 reference